SCHEMBL181775

SCHEMBL181775

CC(C)(C)OC(=O)N[C@@H](CCc1ccccc1)C(=O)O

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.71
CTSS P25774 5/20 0.71
PPARA Q07869 5/20 0.62
PPARG P37231 4/20 0.62
ACE P12821 1/20 0.60
CTSB P07858 2/20 0.56
CTSL P07711 1/20 0.56
PPARD Q03181 2/20 0.56
ATM Q13315 1/20 0.52
IDO1 P14902 1/20 0.51
APP P05067 1/20 0.51
SCN9A Q15858 1/20 0.51
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL181807 1.00 CTSK (0.71) CTSKCTSSPPARAPPARGACE
SCHEMBL181808 1.00 CTSK (0.71) CTSKCTSSPPARAPPARGACE
SCHEMBL8238590 0.95 PPARA (0.70) CTSKCTSSPPARAPPARGACE
SCHEMBL13744253 0.95 PPARA (0.70) CTSKCTSSPPARAPPARGACE
SCHEMBL344068 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL22651626 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL19605638 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL2781406 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL1374859 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL346311 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 473 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180298056-A1 PROCESS FOR THE PREPARATION OF (2S)-N-((S)-1-((S)-4-METHYL-1-((R)-2-METHYL OXIRAN-2-YL)-1-OXOPENTAN-2-YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2-MORPHOLINO ACETAMIDO)-4-PHENYLBUTANAMIDO)-4-METHYLPENTANAMIDE MSN LABORATORIES PRIVATE LIMITED (IN) 2018-10-18 US claimed
WO-2016170544-A1 PROCESS FOR THE PREPARATION OF (2S)-N-((S)-1-((S)-4-METHYL-1-((R)-2-METHYL OXIRAN-2-YL)-1-OXOPENTAN-2-YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2-MORPHOLINO ACETAMIDO)-4-PHENYLBUTANAMIDO)-4-METHYLPENTANAMIDE MSN LABORATORIES PRIVATE LIMITED (IN) 2016-10-27 WO claimed
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2026-05-07 US disclosed
EP-3788039-B1 FACTOR XIIA INHIBITORS UNIV LEEDS INNOVATIONS LTD (GB) 2026-02-11 EP disclosed
US-20260015313-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF PEPTIDREAM INC (JP) 2026-01-15 US disclosed
US-12473331-B2 Macrocyclic compounds as proteasome inhibitors CORNELL UNIVERSITY (US) 2025-11-18 US disclosed
EP-4638415-A1 BIS-ESTER AND AMIDE CATIONIC LIPIDS Sanofi Pasteur Inc. (US) 2025-10-29 EP disclosed
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-09-16 US disclosed
US-12383560-B2 Compounds and uses thereof FOGHORN THERAPEUTICS INC. (US) 2025-08-12 US disclosed
US-12336991-B2 Factor XIIA inhibitors UNIVERSITY OF LEEDS (GB) 2025-06-24 US disclosed
EP-4534524-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF PeptiDream Inc. (JP) 2025-04-09 EP disclosed
US-5153226-A Administering as anticholesterol agents, for atherosclerosis WARNER-LAMBERT COMPANY (US) 1992-10-06 US disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed
US-5149795-A Fungicides BAYER AG (DE) 1992-09-22 US disclosed
EP-0478362-A2 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1992-04-01 EP disclosed
US-5019560-A Method for treating fungal infections with nikkomycin derivatives BAYER AG (DE) 1991-05-28 US disclosed
EP-0415413-A1 Acat inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-06 EP disclosed
EP-0367954-A1 Nikkomycin derivatives, antimycotic compositions of nikkomycin derivatives and azole antimycotics BAYER AG (DE) 1990-05-16 EP disclosed
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed
EP-0352000-A2 Retroviral protease binding peptides SMITHKLINE BEECHAM CORPORATION (US) 1990-01-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SLC26A4, SLC26A3 CTSK 4042/4885CTSS 3662/4885PPARA 2634/4885
US-20260015313-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF NSUN3, BCAT1, SLC43A1 CTSK 4661/4885CTSS 4022/4885PPARA 2794/4885
US-12383560-B2 Compounds and uses thereof VHL, CLN6, TFEB CTSK 2434/4885CTSS 2010/4885PPARA 1483/4885
US-20180298056-A1 PROCESS FOR THE PREPARATION OF (2S)-N-((S)-1-((S)-4-METHYL-1-((R)-2-METHYL OXIRAN-2-YL)-1-OXOPENTAN-2-YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2-MORPHOLINO ACETAMIDO)-4-PHENYLBUTANAMIDO)-4-METHYLPENTANAMIDE OPRL1, OPRM1, ADRA1D CTSK 4506/4885CTSS 3324/4885PPARA 3374/4885
US-12473331-B2 Macrocyclic compounds as proteasome inhibitors PSMB5, PSMB1, PSMB3 CTSK 1101/4885CTSS 640/4885PPARA 4669/4885
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SCNN1G CTSK 2963/4885CTSS 3812/4885PPARA 4410/4885
US-12336991-B2 Factor XIIA inhibitors F11, F13B, F12 CTSK 303/4885CTSS 714/4885PPARA 4768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.