SCHEMBL1923910

SCHEMBL1923910

COCOc1ccc(O)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 5/20 0.54
NR5A1 Q13285 1/20 0.50
APP P05067 2/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
PTGS1 P23219 1/20 0.48
SLC6A2 P23975 1/20 0.48
CYP2C19 P33261 1/20 0.48
PTGS2 P35354 1/20 0.48
SLC6A3 Q01959 1/20 0.48
HIF1A Q16665 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ESR2 Q92731 2/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ESR1 P03372 1/20 0.46
CALM1 P0DP23 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3418462 0.94 ESR2 (0.59) LTA4HNR5A1APPLMNACYP1A2
SCHEMBL9149725 0.90 ALOX15 (0.50) LTA4HNR5A1APPLMNACYP1A2
SCHEMBL3589633 0.87 NQO1 (0.50) LTA4HAPP
SCHEMBL25124165 0.87 ESR1 (0.57) LTA4HNR5A1LMNACYP1A2SLC6A2
SCHEMBL14227001 0.85 PKM (0.66) LTA4HLMNAKMT2A
SCHEMBL8452874 0.85 LTA4H (0.56) LTA4HNR5A1APPLMNACYP1A2
SCHEMBL4599599 0.83 LTA4H (0.48) LTA4HNR5A1APPLMNACYP1A2
SCHEMBL14514637 0.80 CA1 (0.58) APP
SCHEMBL197283 0.80 FYN (0.45) CYP1A2CYP2C19ESR2
SCHEMBL12926336 0.80 MMP2 (0.51) LTA4HCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570648-B2 6,7-dihydro-5H-pyrido[2,3-c]pyridazine derivatives and related compounds as Bcl-xL protein inhibitors and pro-apoptotic agents for treating cancer LES LABORATOIRES SERVIER (FR) 2026-03-10 US disclosed
US-20250215010-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS VASA THERAPEUTICS SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA (PL) 2025-07-03 US disclosed
WO-2025096495-A1 ARYL FLUOROSULFATE-BASED INHIBITORS AS NOVEL ANTITUBERCULAR AGENTS THE SCRIPPS RESEARCH INSTITUTE (US) 2025-05-08 WO disclosed
CN-119923399-A Useful as matrix metalloproteinase inhibitors diazabicyclooctane derivatives of (a) 瓦萨治疗有限责任公司 2025-05-02 CN disclosed
US-12258355-B2 Probes for imaging huntingtin protein CHDI FOUNDATION, INC. (US) 2025-03-25 US disclosed
EP-4499647-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS Vasa Therapeutics Spolka Z Orgraniczona Odpowiedzialnoscia (PL) 2025-02-05 EP disclosed
CN-114450284-B 6, 7-Dihydro-5H-pyrido [2,3-C ] pyridazine derivatives as BCL-XL protein inhibitors 法国施维雅药厂 2024-05-07 CN disclosed
EP-4003989-B1 6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER SERVIER LAB (FR) 2023-12-27 EP disclosed
WO-2023187670-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS VASA THERAPEUTICS SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA (PL) 2023-10-05 WO disclosed
CN-116655618-A Probes for imaging huntingtin CHDI基金会股份有限公司 2023-08-29 CN disclosed
US-20040171634-A1 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use AGOURON PHARMACEUTICALS, LLC 2004-09-02 US disclosed
US-6534524-B1 Antiproliferative agents, including axitinib AGOURON PHARMACEUTICALS, INC. 2003-03-18 US disclosed
US-6531491-B1 Methods of treating cancer and other disease states associated with unwanted angiogenesis and/or cellular proliferation, such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis, and psoriasis, AGOURON PHARAMACEUTICALS, INC. 2003-03-11 US disclosed
EP-1218348-A2 INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEIN KINASES, AND METHODS FOR THEIR USE AGOURON PHARMACEUTICALS, INC. (US) 2002-07-03 EP disclosed
WO-2001002369-A2 INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEIN KINASES, AND METHODS FOR THEIR USE AGOURON PHARMACEUTICALS, INC. (US) 2001-01-11 WO disclosed
US-5932196-A DEOXYARBUTIN DERIVATIVES, STORAGE STABILITY THE PROCTER & GAMBLE COMPANY (US) 1999-08-03 US disclosed
US-5250690-A Selective killing of grassy weeds DOWELANCO (US) 1993-10-05 US disclosed
US-4968343-A GRASSY WEEDS IN PRESENCE OF CORN PLANTS THE DOW CHEMICAL COMPANY (US) 1990-11-06 US disclosed
EP-0205821-A1 Haloalkoxy anilide derivatives of 2-(4-heterocyclic oxyphenoxy)-alkanoic acids and their use as herbicides THE DOW CHEMICAL COMPANY (US) 1986-12-30 EP disclosed
CN-86103114-A The halogenated alkoxy benzene of 2-(4-heterocyclic oxy group phenoxy group) alkanoic acid is for the preparation of amide derivatives and as herbicide applications 1986-12-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040171634-A1 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use CDK3, BRAF, ROCK1 LTA4H 2924/4885NR5A1 1753/4885APP 2058/4885
US-12570648-B2 6,7-dihydro-5H-pyrido[2,3-c]pyridazine derivatives and related compounds as Bcl-xL protein inhibitors and pro-apoptotic agents for treating cancer BCOR, BCL2A1, BAK1 LTA4H 1008/4885NR5A1 430/4885APP 2733/4885
US-20250215010-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS MMP1, MMP9, MMP8 LTA4H 603/4885NR5A1 1965/4885APP 4612/4885
US-12258355-B2 Probes for imaging huntingtin protein HTT, HYPK, HSPBP1 LTA4H 4799/4885NR5A1 2929/4885APP 270/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.