SCHEMBL1977066

SCHEMBL1977066

O=C(Cl)Oc1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
ALOX15 P16050 1/20 0.48
FAAH O00519 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 1/20 0.46
PARP10 Q53GL7 1/20 0.44
CXCL8 P10145 1/20 0.44
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 2/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
GAA P10253 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
HPGD P15428 1/20 0.40
NPC1 O15118 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5696260 0.84 SERPINE1 (0.43) ALDH1A1ALOX15SMN1; SMN2MAPTKDM4E
SCHEMBL30524282 0.84 SERPINE1 (0.43) ALDH1A1ALOX15SMN1; SMN2MAPTKDM4E
SCHEMBL18697277 0.82 FAAH (0.49) ALDH1A1ALOX15FAAHSMN1; SMN2MAPT
SCHEMBL29585912 0.82 FAAH (0.49) ALDH1A1ALOX15FAAHSMN1; SMN2MAPT
SCHEMBL57243 0.82 FAAH (0.49) ALDH1A1ALOX15FAAHSMN1; SMN2MAPT
SCHEMBL2940941 0.82 FAAH (0.49) ALDH1A1ALOX15FAAHSMN1; SMN2MAPT
SCHEMBL6966435 0.80 FAAH (0.47) ALDH1A1ALOX15FAAHSMN1; SMN2MAPT
SCHEMBL57244 0.80 FAAH (0.51) ALDH1A1FAAHSMN1; SMN2MAPTPARP10
SCHEMBL2830676 0.79 CES2 (0.45) FAAHMAPTKDM4EKMT2ACES2
SCHEMBL2322496 0.78 PARP10 (0.53) ALDH1A1FAAHSMN1; SMN2MAPTPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4654968-A1 PROCESS FOR THE PREPARATION OF TIVOZANIB OR A SALT THEREOF Alivus Life Sciences Limited (IN) 2025-12-03 EP disclosed
WO-2024157170-A1 PROCESS FOR THE PREPARATION OF TIVOZANIB OR A SALT THEREOF GLENMARK LIFE SCIENCES LIMITED (IN) 2024-08-02 WO disclosed
CN-116940576-A Method for producing S, S- (6-methylquinoxaline-2, 3-diyl) dithiocarbonate 株式会社大阪曹达 2023-10-24 CN disclosed
WO-2023154344-A1 2-METHYL-4',5'-DIHYDROSPIRO[PIPERIDINE-4,7'-THIENO[2,3-C]PYRAN] DERIVATIVES AS INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed
WO-2022202643-A1 METHOD FOR PRODUCING S,S-(6-METHYLQUINOXALINE-2,3-DIYL)DITHIOCARBONATE 株式会社大阪ソーダ 2022-09-29 WO disclosed
US-10035790-B2 RORγ modulators EXELIXIS, INC. (US) 2018-07-31 US disclosed
US-9346786-B2 Pyrrolidine compounds HOFFMANN-LA ROCHE INC. (US) 2016-05-24 US disclosed
US-9226916-B2 Pyrrolidine derivatives HOFFMANN-LA ROCHE INC. (US) 2016-01-05 US disclosed
US-20150266856-A1 RORGamma Modulators EXELIXIS, INC. 2015-09-24 US disclosed
EP-2513084-B1 PYRROLIDINE DERIVATIVES AS NK-3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2015-07-22 EP disclosed
US-7276511-B2 Benzylamine derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 2007-10-02 US disclosed
US-7276511-B2 Benzylamine derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 2007-10-02 US disclosed
US-20060194841-A1 E.g., N-{2-(3,4-dichlorophenyl)-2-[(3,3-diphenylpropionyl)-methylamino]-4-{spiro[benzo(c)thiophene-1(3H),4'-piperidine]-(2S)-oxide}-1'-yl-butyl}-3,3,3-trifluoro-N-methyl-propionamide hydrochloride, NK-1 or NK-2 receptor antagonists; irritable bowel syndrome, pain, anxiety, COPD, headaches and vomiting ZERIA PHARMACEUTICAL CO., LTD. (JP) 2006-08-31 US disclosed
EP-1650189-A1 BENZYLAMINE DERIVATIVE Zeria Pharmaceutical Co., Ltd. (JP) 2006-04-26 EP disclosed
US-20020082254-A1 Compounds for treating disorders where a decreased level of plasma FFA is desired NOVO NORDISK A/S (DK) 2002-06-27 US disclosed
WO-2001087843-A1 COMPOUNDS FOR TREATING DISORDERS WHERE A DECREASED LEVEL OF PLASMA FFA IS DESIRED NOVO NORDISK A/S (DK) 2001-11-22 WO disclosed
US-5843983-A Diphenylethane compounds containing a saturated heterocyclic group, their preparation, and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1998-12-01 US disclosed
US-5811424-A CONTROL OF DOWNY MILDEW, LATE BLIGHT KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1998-09-22 US disclosed
EP-0790235-A1 Diaryl alkane derivatives containing an alicyclic group, their preparation and their therapeutic and prophylactic uses SANKYO COMPANY LIMITED (JP) 1997-08-20 EP disclosed
US-4376731-A 2-NITRILES THEREOF BOEHRINGER MANNHEIM GMBH (DE) 1983-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150266856-A1 RORGamma Modulators RORB, RORA, RORC ALDH1A1 1877/4885ALOX15 2259/4885FAAH 3398/4885
US-10035790-B2 RORγ modulators RORB, RORA, RORC ALDH1A1 1669/4885ALOX15 1003/4885FAAH 3187/4885
US-20060194841-A1 E.g., N-{2-(3,4-dichlorophenyl)-2-[(3,3-diphenylpropionyl)-methylamino]-4-{spiro[benzo(c)thiophene-1(3H),4'-piperidine]-(2S)-oxide}-1'-yl-butyl}-3,3,3-trifluoro-N-methyl-propionamide hydrochloride, NK-1 or NK-2 receptor antagonists; irritable bowel syndrome, pain, anxiety, COPD, headaches and vomiting KCNAB1, BDKRB2, ARRB1 ALDH1A1 1065/4885ALOX15 2584/4885FAAH 942/4885
US-20020082254-A1 Compounds for treating disorders where a decreased level of plasma FFA is desired FABP1, FFAR2, FFAR1 ALDH1A1 779/4885ALOX15 103/4885FAAH 124/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.