SCHEMBL19856933

SCHEMBL19856933

Cc1ccc(C(=O)N2C[C@@H]3C[C@H]2CN3C(=O)[C@@H](n2c(C(N)=O)cc3ccccc32)C(C)(C)C)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CCR2 P41597 1/20 0.33
NOD2 Q9HC29 3/20 0.32
NOD1 Q9Y239 3/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
PKM P14618 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
TNF P01375 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SPR P35270 1/20 0.30
AVPR2 P30518 1/20 0.30
AVPR1A P37288 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856941 0.94 TNF (0.37) CCR2NOD2NOD1RAB9ATNF
SCHEMBL19856992 0.92 CCR2 (0.34) ALDH1A1CCR2SPRHSD11B1
SCHEMBL19856957 0.91 AVPR1A (0.34) CCR2AVPR2AVPR1AHSD11B1
SCHEMBL19856907 0.91 HCRTR1 (0.33) NOD2NOD1HCRTR1HCRTR2SMN1; SMN2
SCHEMBL19856975 0.90 SMN1; SMN2 (0.34) ALDH1A1CCR2NPC1RAB9APKM
SCHEMBL19856993 0.90 PLA2G10 (0.38) CCR2HCRTR1HCRTR2
SCHEMBL19856929 0.89 CCR2 (0.35) CCR2HCRTR1HCRTR2HSD11B1
SCHEMBL19856988 0.89 NOD2 (0.41) ALDH1A1NOD2NOD1NPC1RAB9A
SCHEMBL19857030 0.85 PLA2G10 (0.38) CCR2HCRTR1HCRTR2
SCHEMBL19856960 0.85 PLA2G10 (0.38) CCR2NOD2NOD1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925857-B1 USE OF TRPV4 ANTAGONISTS TO AMELIORATE HYDROCEPHALUS AND RELATED MATERIALS AND METHODS UNIV INDIANA RES & TECH CORP (US) 2018-02-14 EP claimed