SCHEMBL19860062

SCHEMBL19860062

COC(=O)c1cccc(CCC(=O)Nc2ccc3cnccc3c2)c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
HPGD P15428 1/20 0.61
NOTUM Q6P988 5/20 0.55
ROCK2 O75116 4/20 0.55
LMNA P02545 1/20 0.53
PRMT3 O60678 2/20 0.52
IMPDH2 P12268 3/20 0.51
MAPT P10636 1/20 0.50
CYP4F2 P78329 1/20 0.49
CYP4A11 Q02928 1/20 0.49
RAB9A P51151 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860120 0.89 PRMT3 (0.53) ALDH1A1HPGDNOTUMROCK2PRMT3
SCHEMBL19860064 0.87 PRMT3 (0.54) NOTUMROCK2LMNAPRMT3IMPDH2
SCHEMBL19860067 0.87 PRMT3 (0.54) NOTUMROCK2PRMT3IMPDH2
SCHEMBL3587855 0.83 NOTUM (0.55) ALDH1A1HPGDNOTUMROCK2LMNA
SCHEMBL3566775 0.83 PRMT3 (0.72) NOTUMROCK2LMNAPRMT3IMPDH2
SCHEMBL19860066 0.82 IMPDH2 (0.65) NOTUMLMNAPRMT3IMPDH2MAPT
SCHEMBL19860079 0.82 ALDH1A1 (0.61) ALDH1A1NOTUMROCK2PRMT3IMPDH2
SCHEMBL2164137 0.81 PRMT3 (0.69) NOTUMROCK2LMNAPRMT3IMPDH2
SCHEMBL19860091 0.80 ROCK2 (0.60) NOTUMROCK2PRMT3IMPDH2
SCHEMBL19860089 0.80 ROCK2 (0.55) ALDH1A1NOTUMROCK2LMNAPRMT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed