SCHEMBL19860079

SCHEMBL19860079

CN(C)c1cccc(CCC(=O)Nc2ccc3cnccc3c2)c1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
GAA P10253 1/20 0.61
ALOX15 P16050 1/20 0.61
NOTUM Q6P988 4/20 0.53
PRMT3 O60678 4/20 0.53
IMPDH2 P12268 4/20 0.52
ROCK2 O75116 4/20 0.51
ROCK1 Q13464 2/20 0.48
PLAU P00749 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3566775 0.84 PRMT3 (0.72) GAANOTUMPRMT3IMPDH2ROCK2
SCHEMBL19860064 0.82 PRMT3 (0.54) NOTUMPRMT3IMPDH2ROCK2ROCK1
SCHEMBL19860062 0.82 ALDH1A1 (0.61) ALDH1A1NOTUMPRMT3IMPDH2ROCK2
SCHEMBL2164137 0.82 PRMT3 (0.69) GAANOTUMPRMT3IMPDH2ROCK2
SCHEMBL19860067 0.81 PRMT3 (0.54) NOTUMPRMT3IMPDH2ROCK2ROCK1
SCHEMBL19860091 0.80 ROCK2 (0.60) NOTUMPRMT3IMPDH2ROCK2
SCHEMBL19860089 0.80 ROCK2 (0.55) ALDH1A1NOTUMPRMT3IMPDH2ROCK2
SCHEMBL14124306 0.77 PRMT3 (0.66) GAANOTUMPRMT3IMPDH2ROCK2
SCHEMBL21430054 0.77 IMPDH2 (0.62) NOTUMPRMT3IMPDH2ROCK2ROCK1
SCHEMBL16634909 0.77 PRMT3 (0.61) ALDH1A1NOTUMPRMT3IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed