SCHEMBL19860089

SCHEMBL19860089

N#Cc1cccc(CCC(=O)Nc2ccc3cnccc3c2)c1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.55
PRMT3 O60678 2/20 0.53
IMPDH2 P12268 4/20 0.52
NOTUM Q6P988 4/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 3/20 0.48
MAPK1 P28482 1/20 0.46
ROCK1 Q13464 1/20 0.46
PLAU P00749 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3566775 0.84 PRMT3 (0.72) ROCK2PRMT3IMPDH2NOTUMLMNA
SCHEMBL3594155 0.83 ALDH1A1 (0.58) ROCK2PRMT3IMPDH2NOTUMALDH1A1
SCHEMBL2164137 0.82 PRMT3 (0.69) ROCK2PRMT3IMPDH2NOTUMLMNA
SCHEMBL19860067 0.81 PRMT3 (0.54) ROCK2PRMT3IMPDH2NOTUMROCK1
SCHEMBL19860091 0.80 ROCK2 (0.60) ROCK2PRMT3IMPDH2NOTUM
SCHEMBL19860079 0.80 ALDH1A1 (0.61) ROCK2PRMT3IMPDH2NOTUMALDH1A1
SCHEMBL19860062 0.80 ALDH1A1 (0.61) ROCK2PRMT3IMPDH2NOTUMALDH1A1
SCHEMBL19860064 0.80 PRMT3 (0.54) ROCK2PRMT3IMPDH2NOTUMLMNA
SCHEMBL14124306 0.77 PRMT3 (0.66) ROCK2PRMT3IMPDH2NOTUMLMNA
SCHEMBL21430054 0.77 IMPDH2 (0.62) ROCK2PRMT3IMPDH2NOTUMROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed