SCHEMBL20003227

SCHEMBL20003227

CC(=O)N1CCN(C(=O)N2CC[C@H](Sc3ccc(P)cc3)C2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
CCR5 P51681 1/20 0.36
QDPR P09417 2/20 0.35
KCNH2 Q12809 3/20 0.33
HRH3 Q9Y5N1 2/20 0.33
MCHR1 Q99705 1/20 0.33
MAPT P10636 1/20 0.33
GCK P35557 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BRD4 O60885 1/20 0.32
CASP6 P55212 1/20 0.32
GFER P55789 1/20 0.32
IDO1 P14902 1/20 0.32
ESR1 P03372 1/20 0.32
CHRM1 P11229 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC29A1 Q99808 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002936 0.87 CCR5 (0.46) KMT2ACCR5KCNH2MAPTSMN1; SMN2
SCHEMBL20002407 0.77 SMN1; SMN2 (0.41) KMT2ACCR5SMN1; SMN2KDM1AMAOB
SCHEMBL20002879 0.75 NPC1 (0.44) KMT2ACCR5KCNH2HRH3SMN1; SMN2
SCHEMBL20003224 0.75 KMT2A (0.43) KMT2ASMN1; SMN2
SCHEMBL20002255 0.73 CCR5 (0.49) KMT2ACCR5
SCHEMBL20002297 0.72 NOTUM (0.47) KMT2ACCR5MAPT
SCHEMBL20002294 0.71 PTPN11 (0.36) KMT2ACCR5CHRM1
SCHEMBL20002612 0.70 RORC (0.36) KMT2ACCR5
SCHEMBL20003024 0.69 NOTUM (0.44) KMT2ACCR5MAPT
SCHEMBL20002327 0.69 MAOA (0.45) KMT2AMAPTMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed