SCHEMBL20042797

SCHEMBL20042797

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)n1ccnc1)C2

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
ALDH1A1 P00352 1/20 0.42
FAAH O00519 3/20 0.37
MGLL Q99685 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.34
NR4A1 P22736 1/20 0.34
P2RX7 Q99572 3/20 0.33
MTOR P42345 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.31
GBA1 P04062 1/20 0.30
ACACA Q13085 1/20 0.30
CHRM4 P08173 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042791 0.80 SMN1; SMN2 (0.37) LMNAALDH1A1SMN1; SMN2TSHRNR4A1
SCHEMBL20042804 0.79 ALDH1A1 (0.40) LMNAALDH1A1SMN1; SMN2TSHRNR4A1
SCHEMBL20042786 0.77 LMNA (0.36) LMNAALDH1A1FAAHMGLLSMN1; SMN2
SCHEMBL20042870 0.76 KDM4E (0.35) LMNAALDH1A1SMN1; SMN2TSHRNR4A1
SCHEMBL20042776 0.76 P2RX7 (0.41) LMNASMN1; SMN2TSHRNR4A1P2RX7
SCHEMBL20042832 0.76 CFTR (0.45) LMNAALDH1A1SMN1; SMN2P2RX7KDM4E
SCHEMBL20042839 0.75 P2RX7 (0.45) ALDH1A1SMN1; SMN2TSHRP2RX7MTOR
SCHEMBL20042743 0.75 P2RX7 (0.40) SMN1; SMN2TSHRP2RX7MTORKDM4E
SCHEMBL20042817 0.75 PKM (0.44) LMNAALDH1A1P2RX7KDM4EGBA1
SCHEMBL20042866 0.75 NPY5R (0.33) SMN1; SMN2MTORKDM4ECHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed