SCHEMBL2221471

SCHEMBL2221471

C[Si](C)(C)CCOCn1ccc(C=O)n1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3496820 0.81 DGAT1 (0.35) NPC1DGAT1
SCHEMBL29953218 0.77
SCHEMBL19992397 0.77 NPC1 (0.32) NPC1DGAT1
SCHEMBL31308722 0.76 DGAT1 (0.35) NPC1DGAT1
SCHEMBL20744490 0.76 DGAT1 (0.40) NPC1DGAT1
SCHEMBL30789772 0.76 DGAT1 (0.33) NPC1DGAT1
SCHEMBL401354 0.76 ALDH1A1 (0.39) NPC1DGAT1
SCHEMBL3389626 0.76 DGAT1 (0.32) NPC1DGAT1
SCHEMBL8257898 0.76 P2RX7 (0.35) DGAT1
SCHEMBL31741697 0.75 DGAT1 (0.32) NPC1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116881-A1 KIF MODULATOR COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS INC (US) 2026-04-30 US disclosed
US-20250144093-A1 PYRUVATE KINASE ACTIVATORS FOR USE IN TREATING BLOOD DISORDERS AGIOS PHARMACEUTICALS, INC. 2025-05-08 US disclosed
US-12133853-B2 Pyruvate kinase activators for use in treating blood disorders AGIOS PHARMACEUTICALS, INC. (US) 2024-11-05 US disclosed
WO-2024178390-A1 COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2024-08-29 WO disclosed
US-11957680-B2 Pyruvate kinase activators for use in treating blood disorders AGIOS PHARMACEUTICALS, INC. (US) 2024-04-16 US disclosed
US-11872225-B2 Pyruvate kinase modulators and use thereof AGIOS PHARMACEUTICALS, INC. (US) 2024-01-16 US disclosed
US-11872225-B2 Pyruvate kinase modulators and use thereof AGIOS PHARMACEUTICALS, INC. (US) 2024-01-16 US disclosed
US-11872225-B2 Pyruvate kinase modulators and use thereof AGIOS PHARMACEUTICALS, INC. (US) 2024-01-16 US disclosed
CN-117186119-A Pyruvate kinase activators for the treatment of hematological disorders 安吉奥斯医药品有限公司 2023-12-08 CN disclosed
EP-3601216-B1 SUBSTITUTED DIHYDROINDENE-4-CARBOXAMIDES AND ANALOGS THEREOF, AND METHODS USING SAME FOR THE TREATMENT OF HEPATITIS B VIRUS INFECTION ARBUTUS BIOPHARMA CORP (CA) 2023-10-25 EP disclosed
US-8722686-B2 Hydroxamic acid derivatives useful as antibacterial agents PFIZER INC. (US) 2014-05-13 US disclosed
US-8722686-B2 Hydroxamic acid derivatives useful as antibacterial agents PFIZER INC. (US) 2014-05-13 US disclosed
US-20110178042-A1 Hydroxamic Acid Derivatives Useful as Antibacterial Agents PFIZER INC. (US) 2011-07-21 US disclosed
US-20110178042-A1 Hydroxamic Acid Derivatives Useful as Antibacterial Agents PFIZER INC. (US) 2011-07-21 US disclosed
US-7635703-B2 Imidazole substituted pyrazole kinase inhibitors JANSSEN PHARMACEUTICA N.V. (BE) 2009-12-22 US disclosed
US-20080103172-A1 IMIDAZOLE SUBSTITUTED PYRAZOLE KINASE INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-05-01 US disclosed
WO-2008048503-A2 IMIDAZOLE SUBSTITURED PYRAZOLE KINASE INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-04-24 WO disclosed
US-20070275954-A1 Novel Fused Heterocycles and Uses Thereof ASTRAZENECA AB (SE) 2007-11-29 US disclosed
EP-1751119-A1 NOVEL FUSED HETEROCYCLES AND USES THEREOF AstraZeneca AB (SE) 2007-02-14 EP disclosed
WO-2005111001-A1 NOVEL FUSED HETEROCYCLES AND USES THEREOF ASTRAZENECA AB (SE) 2005-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260116881-A1 KIF MODULATOR COMPOUNDS AND METHODS OF USE KIF2C, KIF5B, KIF5C NPC1 107/4885DGAT1 3064/4885
US-11872225-B2 Pyruvate kinase modulators and use thereof PDK1, PDK2, PDK4 NPC1 3125/4885DGAT1 2745/4885
US-20070275954-A1 Novel Fused Heterocycles and Uses Thereof VIP, CCKBR, HRH2 NPC1 679/4885DGAT1 3316/4885
US-20080103172-A1 IMIDAZOLE SUBSTITUTED PYRAZOLE KINASE INHIBITORS MAP3K19, MAP3K20, MAP3K3 NPC1 2462/4885DGAT1 3840/4885
US-11957680-B2 Pyruvate kinase activators for use in treating blood disorders PDK1, PDK2, PDK3 NPC1 1348/4885DGAT1 2658/4885
US-20110178042-A1 Hydroxamic Acid Derivatives Useful as Antibacterial Agents HCAR1, HDAC1, H1-0 NPC1 2166/4885DGAT1 3136/4885
US-12133853-B2 Pyruvate kinase activators for use in treating blood disorders PDK1, PDK2, PDK3 NPC1 2102/4885DGAT1 3106/4885
US-20250144093-A1 PYRUVATE KINASE ACTIVATORS FOR USE IN TREATING BLOOD DISORDERS PDK1, PDK2, PDK3 NPC1 2102/4885DGAT1 3106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.