SCHEMBL2229145

SCHEMBL2229145

CC1(C)OB(c2ccc3c(c2)-c2cccc4cccc-3c24)OC1(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 12/20 0.48
LPL P06858 11/20 0.48
ALDH1A1 P00352 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CASP1 P29466 2/20 0.43
CASP7 P55210 2/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
HIF1A Q16665 1/20 0.43
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.40
TYMS P04818 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
F11 P03951 1/20 0.37
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18820580 0.90 LIPG (0.40) LIPGLPLALDH1A1TSHRMAPK1
SCHEMBL25223314 0.88 LIPG (0.61) LIPGLPLALDH1A1TSHRMAPK1
SCHEMBL24654439 0.87 LIPG (0.49) LIPGLPLALDH1A1TSHRMAPK1
SCHEMBL16581306 0.87 LPL (0.56) LIPGLPLIRAK4CA1CA2
SCHEMBL2228128 0.86 LPL (0.49) LIPGLPLALDH1A1TSHRMAPK1
SCHEMBL21368178 0.84 LPL (0.40) LIPGLPLALDH1A1TSHRMAPK1
SCHEMBL12200531 0.82 LIPG (0.40) LIPGLPLIRAK4CA1CA2
SCHEMBL19120001 0.81 LIPG (0.43) LIPGLPLIRAK4TYMSCA1
SCHEMBL31062339 0.81 KDM4E (0.51) LIPGLPLMAPK1ATMIRAK4
SCHEMBL17776257 0.81 KDM4E (0.51) LIPGLPLMAPK1ATMIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3368520-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2023-04-26 EP disclosed
US-11355714-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2022-06-07 US disclosed
US-11302870-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2022-04-12 US disclosed
US-20190288206-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2019-09-19 US disclosed
US-20190058133-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2019-02-21 US disclosed
WO-2017071791-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2017-05-04 WO disclosed
US-20160141506-A1 NAPHTHO[2,1-b]FLUORANTHENE COMPOUND, ORGANIC LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, LIGHTING APPARATUS, IMAGE FORMING APPARATUS, AND EXPOSING APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-05-19 US disclosed
US-20160141506-A1 NAPHTHO[2,1-b]FLUORANTHENE COMPOUND, ORGANIC LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, LIGHTING APPARATUS, IMAGE FORMING APPARATUS, AND EXPOSING APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-05-19 US disclosed
US-8026664-B2 Compound and organic light emitting device CANON KABUSHIKI KAISHA (JP) 2011-09-27 US disclosed
US-7977869-B2 Organic luminescent device and benzo[k]fluoranthene compound CANON KABUSHIKI KAISHA (JP) 2011-07-12 US disclosed
US-20100123390-A1 LIGHT-EMITTING DEVICE, IMAGE DISPLAY APPARATUS, AND NOVEL ORGANIC COMPOUND CANON KABUSHIKI KAISHA (JP) 2010-05-20 US disclosed
US-20100123390-A1 LIGHT-EMITTING DEVICE, IMAGE DISPLAY APPARATUS, AND NOVEL ORGANIC COMPOUND CANON KABUSHIKI KAISHA (JP) 2010-05-20 US disclosed
US-20090278447-A1 ORGANIC LUMINESCENT DEVICE AND BENZO[k]FLUORANTHENE COMPOUND CANON KABUSHIKI KAISHA (JP) 2009-11-12 US disclosed
EP-2049616-A1 ORGANIC LUMINESCENT DEVICE AND BENZO[K]FLUORANTHENE COMPOUND Canon Kabushiki Kaisha (JP) 2009-04-22 EP disclosed
US-20090033210-A1 COMPOUND AND ORGANIC LIGHT EMITTING DEVICE CANON KABUSHIKI KAISHA (JP) 2009-02-05 US disclosed
WO-2008015945-A1 ORGANIC LUMINESCENT DEVICE AND BENZO[k]FLUORANTHENE COMPOUND CANON KABUSHIKI KAISHA (JP) 2008-02-07 WO disclosed
WO-2007123256-A1 COMPOUND AND ORGANIC LIGHT EMITTING DEVICE CANON KABUSHIKI KAISHA (JP) 2007-11-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090033210-A1 COMPOUND AND ORGANIC LIGHT EMITTING DEVICE TRPA1, LEF1, FLI1 LIPG 807/4885LPL 672/4885ALDH1A1 427/4885
US-20100123390-A1 LIGHT-EMITTING DEVICE, IMAGE DISPLAY APPARATUS, AND NOVEL ORGANIC COMPOUND OCIAD1, OCIAD2, OR51E2 LIPG 1422/4885LPL 1190/4885ALDH1A1 163/4885
US-11302870-B2 Materials for electronic devices EFNA1, PNMT, FLNB LIPG 2616/4885LPL 4429/4885ALDH1A1 365/4885
US-11355714-B2 Materials for organic electroluminescent devices SLCO4C1, SLCO2A1, SLCO2B1 LIPG 2734/4885LPL 4054/4885ALDH1A1 1315/4885
US-20090278447-A1 ORGANIC LUMINESCENT DEVICE AND BENZO[k]FLUORANTHENE COMPOUND FOXK1, KCNK10, F10 LIPG 1545/4885LPL 550/4885ALDH1A1 1170/4885
US-20190058133-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES SLCO4C1, SLCO2A1, SLCO2B1 LIPG 2734/4885LPL 4054/4885ALDH1A1 1315/4885
US-20160141506-A1 NAPHTHO[2,1-b]FLUORANTHENE COMPOUND, ORGANIC LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, LIGHTING APPARATUS, IMAGE FORMING APPARATUS, AND EXPOSING APPARATUS NAP1L1, NR0B2, AFF1 LIPG 4444/4885LPL 3761/4885ALDH1A1 479/4885
US-20190288206-A1 MATERIALS FOR ELECTRONIC DEVICES EFNA1, PNMT, FLNB LIPG 2668/4885LPL 4415/4885ALDH1A1 337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.