SCHEMBL22308264

SCHEMBL22308264

BBn1cc(S(=O)(=O)c2ccc(C)cc2)nn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.44
GAA P10253 1/20 0.44
NR1I2 O75469 1/20 0.41
HSP90AA1 P07900 2/20 0.40
NLRP3 Q96P20 1/20 0.40
KMT2A Q03164 3/20 0.38
CXCR5 P32302 1/20 0.38
APLNR P35414 1/20 0.38
RAB9A P51151 1/20 0.38
CCR6 P51684 1/20 0.38
GFER P55789 1/20 0.38
PKM P14618 4/20 0.38
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
RAPGEF4 Q8WZA2 1/20 0.37
HPGD P15428 2/20 0.36
PTGS2 P35354 2/20 0.36
PTGS1 P23219 1/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22308629 0.85 AKR1B1 (0.44) AKR1B1KMT2APKMALDH1A1POLB
SCHEMBL22307381 0.84 AKR1B1 (0.41) AKR1B1KMT2APKMALDH1A1HPGD
SCHEMBL22308428 0.84 ALDH1A1 (0.43) NR1I2KMT2ARAB9AGFERALDH1A1
SCHEMBL22307376 0.81 AGTR1 (0.43) HSP90AA1KMT2ACXCR5APLNRRAB9A
SCHEMBL22307873 0.81 MAOA (0.40) GAANR1I2PKMALDH1A1MAPT
SCHEMBL22308350 0.78 ALDH3A1 (0.34) NR1I2KMT2AGFERPTGS2CA1
SCHEMBL22308585 0.77 L3MBTL1 (0.37) GAAALDH1A1POLBHTTRAPGEF4
SCHEMBL22308263 0.76 GAA (0.48) AKR1B1GAANR1I2HSP90AA1NLRP3
SCHEMBL22308352 0.75 NR1I2 (0.39) AKR1B1GAANR1I2PKMALDH1A1
SCHEMBL14434942 0.74 GAA (0.46) AKR1B1GAANR1I2HSP90AA1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11358940-B2 K-Ras modulators THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-06-14 US disclosed
US-20200247762-A1 K-RAS MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-08-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200247762-A1 K-RAS MODULATORS KRAS, HRAS, NRAS AKR1B1 2660/4885GAA 3688/4885NR1I2 2549/4885
US-11358940-B2 K-Ras modulators KRAS, HRAS, NRAS AKR1B1 1943/4885GAA 3226/4885NR1I2 1591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.