SCHEMBL2273564

SCHEMBL2273564

O=C(Nc1cc(Oc2ccccc2)ccc1C(=O)O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.61
HDAC8 Q9BY41 2/20 0.61
HDAC6 Q9UBN7 2/20 0.61
SERPINE1 P05121 1/20 0.61
PRSS12 P56730 2/20 0.57
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
NPC1 O15118 1/20 0.54
ALDH1A1 P00352 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
KCNH2 Q12809 1/20 0.54
PKM P14618 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
SLC16A3 O15427 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269138 0.90 SERPINE1 (0.57) HDAC1HDAC8HDAC6SERPINE1MEN1
SCHEMBL2272043 0.88 SERPINE1 (0.75) HDAC1HDAC8HDAC6SERPINE1PRSS12
SCHEMBL2294521 0.86 SERPINE1 (0.66) HDAC1HDAC8HDAC6SERPINE1MEN1
SCHEMBL2271588 0.86 SERPINE1 (0.64) SERPINE1MEN1KMT2ANPC1RAB9A
SCHEMBL2270287 0.85 PYGM (0.70) HDAC1HDAC8HDAC6SERPINE1PRSS12
SCHEMBL2275201 0.85 ACLY (0.67) SERPINE1PRSS12MEN1KMT2APKM
SCHEMBL2270621 0.84 GALK1 (0.68) SERPINE1NPC1RAB9A
SCHEMBL2276745 0.84 SERPINE1 (0.65) SERPINE1MEN1KMT2ANPC1RAB9A
SCHEMBL2269563 0.84 STK39 (0.57) SERPINE1PRSS12MEN1KMT2AALDH1A1
SCHEMBL2272347 0.84 SERPINE1 (0.69) SERPINE1MEN1KMT2ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
CN-101094829-A Novel anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO LTD (JP) 2007-12-26 CN disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 HDAC1 71/4885HDAC8 204/4885HDAC6 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.