SCHEMBL2306872

SCHEMBL2306872

ON=C1CCc2cc(Br)ccc21

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.62
SRD5A1 P18405 2/20 0.50
SRD5A2 P31213 1/20 0.50
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP10 Q53GL7 1/20 0.43
PARP11 Q9NR21 1/20 0.43
HPGD P15428 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
BRAF P15056 6/20 0.43
MAPK3 P27361 5/20 0.43
MAPK1 P28482 5/20 0.43
CYP19A1 P11511 6/20 0.41
CYP11B1 P15538 6/20 0.41
CYP11B2 P19099 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2306868 1.00 HTT (0.62) HTTSRD5A1SRD5A2LMNAHSD17B10
SCHEMBL11898554 1.00 HTT (0.62) HTTSRD5A1SRD5A2LMNAHSD17B10
SCHEMBL1809334 0.89 HPGD (0.53) HTTSRD5A1SRD5A2PARP10PARP11
SCHEMBL16621035 0.89 HPGD (0.53) HTTSRD5A1SRD5A2PARP10PARP11
SCHEMBL11971363 0.89 HPGD (0.53) HTTSRD5A1SRD5A2PARP10PARP11
SCHEMBL595554 0.85 HTT (0.49) HTTSRD5A1SRD5A2LMNAHSD17B10
SCHEMBL595553 0.85 HTT (0.49) HTTSRD5A1SRD5A2LMNAHSD17B10
SCHEMBL595555 0.85 HTT (0.49) HTTSRD5A1SRD5A2LMNAHSD17B10
SCHEMBL204100 0.79 SRD5A1 (0.64) SRD5A1SRD5A2PARP10PARP11L3MBTL1
SCHEMBL31268305 0.79 SRD5A1 (0.64) SRD5A1SRD5A2PARP10PARP11L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175272-A Method for preparing R-5-bromo-1-aminoindane WU LING 2015-12-23 CN claimed
CN-105130824-A Method for preparing S-5-bromo-1-aminoindane WU LING 2015-12-09 CN claimed
US-20230255200-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VI BASF SE (DE) 2023-08-17 US disclosed
EP-4178943-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VI BASF SE (DE) 2023-05-17 EP disclosed
CN-115836049-A Use of strobilurin-type compounds to control phytopathogenic fungi containing the amino acid substitution F129L in the mitochondrial cytochrome b protein conferring tolerance to Qo inhibitor VI 巴斯夫欧洲公司 2023-03-21 CN disclosed
EP-3960727-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VI BASF SE (DE) 2022-03-02 EP disclosed
WO-2022008303-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VI BASF SE (DE) 2022-01-13 WO disclosed
US-9809553-B2 Isoquinoline compounds, a process for their preparation, and pharmaceutical compositions containing them LES LABORATOIRES SERVIER (FR) 2017-11-07 US disclosed
US-20170137385-A1 ISOQUINOLINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2017-05-18 US disclosed
EP-3095780-A1 PESTICIDAL ARYLPYRROLIDINES Bayer Intellectual Property GmbH (DE) 2016-11-23 EP disclosed
US-9271499-B2 Pesticidal arylpyrrolidines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-03-01 US disclosed
WO-2010043315-A1 PESTICIDAL (HETERO) ARYLPYRROLIDINES BAYER CROPSCIENCE AG (DE) 2010-04-22 WO disclosed
US-20090137547-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS HOLDING, INC. 2009-05-28 US disclosed
US-7414142-B2 5-aryl-indan-1-one oximes and analogs useful as progesterone receptor modulators WYETH (US) 2008-08-19 US disclosed
CN-101137414-A Multicyclic bis-amide mmp inhibitors ALANTOS PHARMACEUTICALS INC (US) 2008-03-05 CN disclosed
EP-1843820-A1 MULTICYCLIC BIS-AMIDE MMP INHIBITORS Alantos Pharmaceuticals, Inc. (US) 2007-10-17 EP disclosed
US-20070066637-A1 5-Aryl-indan-1-one oximes and analogs useful as progesterone receptor modulators WYETH (US) 2007-03-22 US disclosed
WO-2006083454-A1 MULTICYCLIC BIS-AMIDE MMP INHIBITORS ALANTOS PHARMACEUTICALS, INC. (US) 2006-08-10 WO disclosed
US-20060173183-A1 Multicyclic bis-amide MMP inhibitors ALANTOS PHARMACEUTICALS, INC., 2006-08-03 US disclosed
WO-1996036596-A1 3,4-DISUBSTITUTED-PHENYLSULPHONAMIDES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173183-A1 Multicyclic bis-amide MMP inhibitors MMP13, MMP3, MMP11 HTT 2111/4885SRD5A1 4641/4885SRD5A2 4656/4885
US-20170137385-A1 ISOQUINOLINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MYLK, MYLK2, MYLK3 HTT 3543/4885SRD5A1 3199/4885SRD5A2 3288/4885
US-20090137547-A1 Heterobicyclic metalloprotease inhibitors MMP13, TIMP3, MMP3 HTT 2315/4885SRD5A1 3637/4885SRD5A2 3698/4885
US-20070066637-A1 5-Aryl-indan-1-one oximes and analogs useful as progesterone receptor modulators CYP19A1, PGR, GNRHR HTT 4288/4885SRD5A1 31/4885SRD5A2 38/4885
US-20230255200-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS VI COX5B, SQOR, COX6B1 HTT 2864/4885SRD5A1 1299/4885SRD5A2 1682/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.