Licofelone

Licofelone

SCHEMBL237833

CC1(C)Cc2c(-c3ccccc3)c(-c3ccc(Cl)cc3)c(CC(=O)O)n2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 1.00
PTGS1 P23219 3/20 1.00
PTGES O14684 2/20 1.00
ALOX5AP P20292 1/20 1.00
PTGS2 P35354 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Licofelone SCHEMBL1843506 0.96 PTGES (0.92) ALOX5PTGS1PTGESALOX5APPTGS2
Licofelone SCHEMBL7737421 0.94 PTGES (0.88) ALOX5PTGS1PTGESALOX5APPTGS2
SCHEMBL9458992 0.93 ALOX5 (0.86) ALOX5PTGS1PTGESALOX5APPTGS2
SCHEMBL5560426 0.92 PTGES (0.85) ALOX5PTGS1PTGESALOX5APPTGS2
SCHEMBL13697422 0.92 PTGES (0.85) ALOX5PTGS1PTGESALOX5APPTGS2
SCHEMBL19499839 0.92 PTGES (0.85) ALOX5PTGS1PTGESALOX5APPTGS2
Licofelone SCHEMBL1394262 0.92 PTGES (0.84) ALOX5PTGS1PTGESALOX5APPTGS2
Licofelone SCHEMBL1393673 0.91 PTGES (0.83) ALOX5PTGS1PTGESALOX5APPTGS2
Licofelone SCHEMBL7738810 0.91 PTGES (0.83) ALOX5PTGS1PTGESALOX5APPTGS2
SCHEMBL4087247 0.91 PTGES (0.83) ALOX5PTGS1PTGESALOX5APPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1106 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260061062-A1 MACROMOLECULAR PRODRUG-BASED THERMOSENSITIVE INJECTABLE GEL AS A NOVEL DRUG DELIVERY PLATFORM UNIV NEBRASKA (US) 2026-03-05 US claimed
US-12545750-B2 Method for the diimide hydrogenation of emulsified unsaturated polymers PARKER DANE K (US) 2026-02-10 US claimed
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
US-20250332143-A1 COMPOSITION COMPRISING ALOX5 INHIBITOR FOR PREVENTING OR TREATING SARCOPENIA PLUTO INC (KR) 2025-10-30 US claimed
WO-2025137653-A1 METHODS AND COMPOSITIONS OF POLYCYCLIC AND A DUAL ACTING NITROXIDE COMPOUNDS FOR TREATMENT OF FAT CELL ASSOCIATED DISEASES MELLICELL, INC. (US) 2025-06-26 WO claimed
CN-119732949-A Use of Licofelone and taxus medicine composition in treating solid tumor 典晶医药(无锡)有限公司 2025-04-01 CN claimed
WO-2025035205-A1 PHARMACEUTICAL COMBINATIONS COMPRISING A SUBSTITUTED THIOPHENE FUSED CYCLOHEXANONE DERIVATIVE AND A CYCLOOXYGENASE (COX) INHIBITOR, AND THEIR USE FOR THE TREATMENT OF PAIN NEURASIC THERAPEUTICS INC. (CA) 2025-02-20 WO claimed
US-20250041275-A1 COMPOSITION FOR USE IN THE TREATMENT OF A DISEASE RAMBAM MED-TECH LTD. (IL) 2025-02-06 US claimed
WO-2005074930-A1 PHARMACEUTICAL COMBINATIONS OF (S) -PANTOPRAZOLE WITH NSAID OR CORTICOSTEROIDS ALTANA PHARMA AG (DE) 2005-08-18 WO claimed
EP-1505964-A1 ANNELATED PYRROLE COMPOUNDS AS PROTON PUMP INHIBITORS FOR TREATING ULCER MERCKLE GMBH (DE) 2005-02-16 EP claimed
US-20050004108-A1 Use of annellated pyrrole compounds in the treatment of articular cartilage or subchondral bone degenaration MERCKLE GMBH (DE) 2005-01-06 US claimed
US-20040242597-A1 Combination NYCOMED GMBH (DE) 2004-12-02 US claimed
WO-2004071391-A2 IMIDAZOPYRIDINES CONTAINING COMBINATIONS AND THEIR USE IN TREATING GASTROINTESTINAL INFLAMMATORY DISORDERS ALTANA PHARMA AG (DE) 2004-08-26 WO claimed
EP-1429807-A2 COMBINATION OF A NSAID AND A PDE-4 INHIBITOR ALTANA Pharma AG (DE) 2004-06-23 EP claimed
EP-1427410-A1 USE OF ANNELLATED PYRROLE COMPOUNDS IN THE TREATMENT OF ARTICULAR CARTILAGE OR SUBCHONDRAL BONE DEGENERATION MERCKLE GMBH (DE) 2004-06-16 EP claimed
WO-2003097041-A1 ANNELATED PYRROLE COMPOUNDS AS PROTON PUMP INHIBITORS FOR TREATING ULCER MERCKLE GMBH (DE) 2003-11-27 WO claimed
WO-2003024489-A2 COMBINATION OF A NSAID AND A PDE-4 INHIBITOR ALTANA PHARMA AG (DE) 2003-03-27 WO claimed
WO-2003020267-A1 USE OF ANNELLATED PYRROLE COMPOUNDS IN THE TREATMENT OF ARTICULAR CARTILAGE OR SUBCHONDRAL BONE DEGENERATION MERCKLE GMBH (DE) 2003-03-13 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260061062-A1 MACROMOLECULAR PRODRUG-BASED THERMOSENSITIVE INJECTABLE GEL AS A NOVEL DRUG DELIVERY PLATFORM CD44, ALG1, HSF1 ALOX5 3180/4885PTGS1 59/4885PTGES 533/4885
US-20250332143-A1 COMPOSITION COMPRISING ALOX5 INHIBITOR FOR PREVENTING OR TREATING SARCOPENIA MYOF, ALOX5, MYLK2 ALOX5 2/4885PTGS1 893/4885PTGES 1682/4885
US-20250041275-A1 COMPOSITION FOR USE IN THE TREATMENT OF A DISEASE SLC10A2, SLC10A1, SLC2A2 ALOX5 179/4885PTGS1 282/4885PTGES 190/4885
US-12545750-B2 Method for the diimide hydrogenation of emulsified unsaturated polymers ALOX15, SOD1, ALOX12 ALOX5 4/4885PTGS1 459/4885PTGES 73/4885
US-20050004108-A1 Use of annellated pyrrole compounds in the treatment of articular cartilage or subchondral bone degenaration BMP4, COL2A1, ACP3 ALOX5 2926/4885PTGS1 88/4885PTGES 710/4885
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ASAH2, ASAH1, GBA2 ALOX5 932/4885PTGS1 1433/4885PTGES 1806/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.