SCHEMBL24066445

SCHEMBL24066445

Cc1ccc(-c2cc(C(C)C)c(C)cn2)cc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.40
USP1 O94782 1/20 0.39
WDR48 Q8TAF3 1/20 0.39
DYRK1A Q13627 2/20 0.38
ALOX5AP P20292 2/20 0.38
FEN1 P39748 2/20 0.38
NPC1 O15118 2/20 0.37
ADORA3 P0DMS8 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
METAP2 P50579 1/20 0.37
ADORA2B P29275 1/20 0.37
KDR P35968 2/20 0.36
CAMKK2 Q96RR4 1/20 0.36
PDGFRB P09619 1/20 0.36
FLT3 P36888 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ENPP3 O14638 1/20 0.35
ENPP1 P22413 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24631952 0.94 LDHA (0.40) LDHAUSP1WDR48DYRK1AALOX5AP
SCHEMBL26262042 0.91 LDHA (0.43) LDHAUSP1WDR48DYRK1AALOX5AP
SCHEMBL18729632 0.88 LDHA (0.50) LDHAUSP1WDR48NPC1KDR
SCHEMBL24066448 0.88 LDHA (0.46) LDHADYRK1AALOX5APFEN1NPC1
SCHEMBL19454850 0.84 LDHA (0.47) LDHADYRK1AALOX5APFEN1NPC1
SCHEMBL26714895 0.84 LDHA (0.41) LDHAUSP1WDR48ALOX5APFEN1
SCHEMBL23562222 0.81 ADORA3 (0.40) LDHAUSP1WDR48DYRK1AALOX5AP
SCHEMBL19373713 0.80 CYP1A2 (0.45) ALOX5APFEN1NPC1METAP2KDR
SCHEMBL22087946 0.79 LDHA (0.45) LDHADYRK1ANPC1ADORA3ADORA2A
SCHEMBL24404662 0.78 LDHA (0.44) LDHADYRK1AALOX5APFEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240074301-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2024-02-29 US disclosed
US-11827651-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-11-28 US disclosed
US-20230371358-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-11-16 US disclosed
US-20230337522-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-19 US disclosed
US-20230337523-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-19 US disclosed
US-20230322829-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-12 US disclosed
US-20230320188-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-10-05 US disclosed
US-20230303601-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-09-28 US disclosed
US-20230287011-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-09-14 US disclosed
US-20230284517-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-09-07 US disclosed
US-11739081-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-08-29 US disclosed
US-20230263048-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-08-17 US disclosed
US-11685754-B2 Heteroleptic organic electroluminescent materials UNIVERSAL DISPLAY CORPORATION (US) 2023-06-27 US disclosed
US-20230143449-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-05-11 US disclosed
US-20230130017-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-04-27 US disclosed
US-20230020526-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2023-01-19 US disclosed
US-20220259242-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2022-08-18 US disclosed
US-20220135606-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2022-05-05 US disclosed
US-20210380617-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2021-12-09 US disclosed
US-20210376261-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2021-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (20 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11685754-B2 Heteroleptic organic electroluminescent materials IK, ORC3, CACNA2D2 LDHA 892/4885USP1 4832/4885WDR48 3738/4885
US-20220135606-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES GLRA3, GLRA2, LIFR LDHA 2081/4885USP1 4570/4885WDR48 3998/4885
US-20230303601-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES MGLL, SELENOI, APOL1 LDHA 1714/4885USP1 4329/4885WDR48 4561/4885
US-20220259242-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES PDCD1LG2, CD274, L1CAM LDHA 408/4885USP1 4156/4885WDR48 3724/4885
US-11739081-B2 Organic electroluminescent materials and devices ICMT, KCNQ2, KCNQ1 LDHA 58/4885USP1 4879/4885WDR48 2877/4885
US-20230284517-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES ICOSLG, OCIAD2, OCIAD1 LDHA 439/4885USP1 2859/4885WDR48 3980/4885
US-20230337522-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES L1CAM, EML4, LBR LDHA 375/4885USP1 4601/4885WDR48 4448/4885
US-20230020526-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES RO60, RPS10, SOD1 LDHA 602/4885USP1 3317/4885WDR48 2611/4885
US-20230320188-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OCIAD2, MLX LDHA 452/4885USP1 4523/4885WDR48 3790/4885
US-20230130017-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OCIAD2, SSB LDHA 257/4885USP1 4689/4885WDR48 3835/4885
US-20230337523-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES LBR, OCIAD1, OCIAD2 LDHA 358/4885USP1 3942/4885WDR48 4325/4885
US-20230287011-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OXGR1, OCIAD1 LDHA 273/4885USP1 4613/4885WDR48 2601/4885
US-20230263048-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OCIAD2, ODC1 LDHA 511/4885USP1 4600/4885WDR48 3255/4885
US-20230143449-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OCIAD1, OXER1 LDHA 707/4885USP1 3901/4885WDR48 3766/4885
US-20240074301-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES ICOSLG, OCIAD2, OSBP LDHA 179/4885USP1 4820/4885WDR48 4625/4885
US-20210376261-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OCIAD1, TPO LDHA 2708/4885USP1 4383/4885WDR48 2474/4885
US-20230322829-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OCIAD1, ICOSLG LDHA 3499/4885USP1 4304/4885WDR48 3432/4885
US-20230371358-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES LIFR, SOD1, ROS1 LDHA 550/4885USP1 2926/4885WDR48 4330/4885
US-11827651-B2 Organic electroluminescent materials and devices SSB, L1CAM, LEF1 LDHA 51/4885USP1 4303/4885WDR48 3389/4885
US-20210380617-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES SOD1, CRKL, ROS1 LDHA 609/4885USP1 4639/4885WDR48 3589/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.