SCHEMBL2464115

SCHEMBL2464115

N#CC=NNc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 2/20 0.52
MAPT P10636 11/20 0.44
GAA P10253 7/20 0.44
ALDH1A1 P00352 6/20 0.44
RAB9A P51151 6/20 0.44
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
HPGD P15428 4/20 0.44
LMNA P02545 3/20 0.44
GFER P55789 1/20 0.44
KDM4E B2RXH2 5/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 2/20 0.39
CYP1A1 P04798 1/20 0.39
TSHR P16473 1/20 0.39
CYP1B1 Q16678 1/20 0.39
SENP7 Q9BQF6 2/20 0.39
SMN1; SMN2 Q16637 5/20 0.38
NPC1 O15118 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2143888 0.79 MAPT (0.46) MAPTGAAALDH1A1RAB9AMEN1
SCHEMBL379196 0.77 MAPT (0.57) MAPTGAAALDH1A1RAB9AMEN1
SCHEMBL3074596 0.75 NOX1 (0.58) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL1005100 0.75 NOX1 (0.58) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL3074599 0.75 NOX1 (0.58) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL16111930 0.74 NOX1 (0.62) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL16111932 0.74 NOX1 (0.62) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL13109406 0.74 NOX1 (0.62) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL11831353 0.73 NOX1 (0.56) NOX1MAPTGAAALDH1A1RAB9A
SCHEMBL11831344 0.73 NOX1 (0.56) NOX1MAPTGAAALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210161937-A1 ACTIVATION OF MITOCHONDRIAL UNCOUPLING AS A THERAPEUTIC INTERVENTION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2021-06-03 US claimed
WO-2019147626-A1 ACTIVATION OF MITOCHONDRIAL UNCOUPLING AS A THERAPEUTIC INTERVENTION THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2019-08-01 WO claimed
US-20260081034-A1 SYSTEMS AND METHODS FOR MEASURING, LEARNING, AND USING EMERGENT PROPERTIES OF COMPLEX ADAPTIVE SYSTEMS EMERJA CORP (US) 2026-03-19 US disclosed
US-20260081035-A1 SYSTEMS AND METHODS FOR MEASURING, LEARNING, AND USING EMERGENT PROPERTIES OF COMPLEX ADAPTIVE SYSTEMS EMERJA CORP (US) 2026-03-19 US disclosed
US-20250382328-A1 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS JENIUS PHARMA LLC (US) 2025-12-18 US disclosed
US-12454549-B2 Treatments for diseases and disorders that involve oxidative stress JENIUS PHARMA, LLC (US) 2025-10-28 US disclosed
US-12312599-B2 Methods, compositions, and kits for producing beige adipocytes and treating metabolic disorders MaineHealth (US) 2025-05-27 US disclosed
EP-4536265-A2 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS Jenius Pharma, LLC (US) 2025-04-16 EP disclosed
US-20240132542-A1 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS Allegro Pharmaceuticals, LLC 2024-04-25 US disclosed
WO-2023239716-A2 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS Allegro Pharmaceuticals, LLC (US) 2023-12-14 WO disclosed
US-20230335287-A1 SYSTEMS AND METHODS FOR MEASURING, LEARNING, AND USING EMERGENT PROPERTIES OF COMPLEX ADAPTIVE SYSTEMS EMERJA CORPORATION 2023-10-19 US disclosed
EP-0511273-A4 LIPOSOMES AS CONTRAST AGENTS FOR ULTRASONIC IMAGING 1993-03-31 EP disclosed
EP-0511273-A1 LIPOSOMES AS CONTRAST AGENTS FOR ULTRASONIC IMAGING IMARX PHARMACEUTICAL CORP. (US) 1992-11-04 EP disclosed
US-5149319-A Methods for providing localized therapeutic heat to biological tissues and fluids CEREVAST THERAPEUTICS, INC. 1992-09-22 US disclosed
US-5123414-A Liposomes as contrast agents for ultrasonic imaging and methods for preparing the same CITIZENS BANK, N.A. 1992-06-23 US disclosed
US-5088499-A Medical diagnosis CITIZENS BANK, N.A. 1992-02-18 US disclosed
WO-1991009629-A1 LIPOSOMES AS CONTRAST AGENTS FOR ULTRASONIC IMAGING UNGER EVAN C (US) 1991-07-11 WO disclosed
EP-0412211-A1 Cancer therapy system THERAPEUTICAL SYSTEMS CORPORATION (US) 1991-02-13 EP disclosed
US-4935450-A Cancer therapy system for effecting oncolysis of malignant neoplasms THERAPEUTICAL SYSTEMS CORPORATION (US) 1990-06-19 US disclosed
US-4724234-A ADMINISTERING NUTRITIONAL REGIMEN AND AGENTS WHICH UNCOUPLE OXIDATIVE PHOSPHORYLATION THERAPEUTICAL SYSTEMS CORP. (US) 1988-02-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240132542-A1 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS GPX4, GPX1, TXNRD2 NOX1 50/4885MAPT 694/4885GAA 174/4885
US-12454549-B2 Treatments for diseases and disorders that involve oxidative stress GPX4, GPX1, TXNRD2 NOX1 50/4885MAPT 694/4885GAA 174/4885
US-20250382328-A1 TREATMENTS FOR DISEASES AND DISORDERS THAT INVOLVE OXIDATIVE STRESS GPX4, GPX1, TXNRD2 NOX1 50/4885MAPT 694/4885GAA 174/4885
US-20260081035-A1 SYSTEMS AND METHODS FOR MEASURING, LEARNING, AND USING EMERGENT PROPERTIES OF COMPLEX ADAPTIVE SYSTEMS PYGB, CRH, CRY1 NOX1 4808/4885MAPT 968/4885GAA 2005/4885
US-12312599-B2 Methods, compositions, and kits for producing beige adipocytes and treating metabolic disorders FABP4, LIPC, PNLIP NOX1 2907/4885MAPT 3885/4885GAA 269/4885
US-20260081034-A1 SYSTEMS AND METHODS FOR MEASURING, LEARNING, AND USING EMERGENT PROPERTIES OF COMPLEX ADAPTIVE SYSTEMS CRH, HCRTR1, PER2 NOX1 4763/4885MAPT 1473/4885GAA 2899/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.