SCHEMBL2486381

SCHEMBL2486381

CCCN[C@H](CCC)Cc1cc2ccccc2o1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.44
CYP2D6 P10635 1/20 0.43
HIF1A Q16665 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
AGXT P21549 1/20 0.41
PSMB5 P28074 2/20 0.40
PSMB8 P28062 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIN1 Q13526 1/20 0.39
HDAC3 O15379 1/20 0.38
ADRA2A P08913 1/20 0.36
HTR1A P08908 3/20 0.36
HTR2B P41595 3/20 0.36
FCER2 P06734 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL398301 1.00 LOXL2 (0.44) LOXL2CYP2D6HIF1AMAOAMAOB
Hydrochloric Acid SCHEMBL2488027 0.99 LOXL2 (0.43) LOXL2CYP2D6HIF1AMAOAMAOB
Hydrochloric Acid SCHEMBL2488414 0.99 LOXL2 (0.43) LOXL2CYP2D6HIF1AMAOAMAOB
Hydrochloric Acid SCHEMBL2488024 0.99 LOXL2 (0.43) LOXL2CYP2D6HIF1AMAOAMAOB
SCHEMBL30457900 0.77 TAS1R3 (0.50) LOXL2AGXTPSMB5PSMB8TAS1R3
SCHEMBL4436085 0.76 CYP2D6 (0.44) LOXL2CYP2D6HIF1AMAOAMAOB
SCHEMBL4340930 0.76 CYP2D6 (0.44) LOXL2CYP2D6HIF1AMAOAMAOB
SCHEMBL19550896 0.74 LOXL2 (0.43) LOXL2CYP2D6HIF1AMAOAMAOB
SCHEMBL30458044 0.74 SIGMAR1 (0.49) LOXL2CYP2D6HIF1AMAOBSIGMAR1
SCHEMBL30457823 0.74 SIGMAR1 (0.49) LOXL2CYP2D6HIF1AMAOBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3226852-B1 ARYLALKYLAMINE COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF CANCER SEMMELWEIS UNIV (HU) 2020-03-18 EP claimed
US-10258599-B2 Compounds for use in the prevention or treatment of cancer SEMMELWEIS UNIVERSITY (HU) 2019-04-16 US claimed
US-20170319535-A1 COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF CANCER SEMMELWEIS UNIVERSITY (HU) 2017-11-09 US claimed
US-20260027148-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS BEXSON BIOMEDICAL INC (US) 2026-01-29 US disclosed
US-20260014191-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS BEXSON BIOMEDICAL INC (US) 2026-01-15 US disclosed
US-20260014190-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS BEXSON BIOMEDICAL INC (US) 2026-01-15 US disclosed
US-12472201-B2 Complexing agent salt formulations of pharmaceutical compounds BEXSON BIOMEDICAL, INC. (US) 2025-11-18 US disclosed
US-20250345458-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL INC (US) 2025-11-13 US disclosed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO disclosed
EP-4525916-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS Bexson Biomedical, Inc. (US) 2025-03-26 EP disclosed
US-20250051778-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS OF USE THEREOF WAVE LIFE SCIENCES LTD. (SG) 2025-02-13 US disclosed
EP-1905760-B1 PROCESS FOR PRODUCTION OF OPTICALLY ACTIVE AMINOPENTANE DERIVATIVE, INTERMEDIATE IN THE PROCESS AND PROCESS FOR PRODUCTION OF THE INTERMEDIATE FUJIMOTO CO LTD (JP) 2011-10-26 EP disclosed
US-20100324300-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE AMINOPENTANE DERIVATIVE, INTERMEDIATE AND PROCESS FOR PREPARING INTERMEDIATE YONEDA FUMIO 2010-12-23 US disclosed
US-7807840-B2 Process for preparing optically active aminopentane derivative, intermediate and process for preparing intermediate FUJIMOTO CO., LTD. (JP) 2010-10-05 US disclosed
EP-2086331-A2 METHODS OF TREATING NEURONAL DISORDERS USING MNTF PEPTIDES AND ANALOGS THEREOF Genervon Biopharmaceuticals LLC (US) 2009-08-12 EP disclosed
US-20090124813-A1 Process for Preparing Optically Active Aminopentane Derivative, Intermediate and Process for Preparing Intermediate FUJIMOTO CO., LTD. (JP) 2009-05-14 US disclosed
US-20090048162-A1 METHODS OF TREATING NEURONAL DISORDERS USING MNTF PEPTIDES AND ANALOGS THEREOF GENERVON BIOPHARMACEUTICALS LLC (US) 2009-02-19 US disclosed
WO-2008057609-A2 METHODS OF TREATING NEURONAL DISORDERS USING MNTF PEPTIDES AND ANALOGS THEREOF GENERVON BIOPHARMACEUTICALS LLC (US) 2008-05-15 WO disclosed
EP-1905760-A1 PROCESS FOR PRODUCTION OF OPTICALLY ACTIVE AMINOPENTANE DERIVATIVE, INTERMEDIATE IN THE PROCESS AND PROCESS FOR PRODUCTION OF THE INTERMEDIATE Fujimoto Co., Ltd. (JP) 2008-04-02 EP disclosed
JP-2003089643-A APOPTOSIS SUPPRESSING AGENT FUJIMOTO CORPORATION:KK 2003-03-28 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090124813-A1 Process for Preparing Optically Active Aminopentane Derivative, Intermediate and Process for Preparing Intermediate API5, CASP5, BAD LOXL2 3348/4885CYP2D6 232/4885HIF1A 3419/4885
US-20260014191-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS SLC6A4, SLC6A3, SIGMAR1 LOXL2 4310/4885CYP2D6 25/4885HIF1A 4630/4885
US-10258599-B2 Compounds for use in the prevention or treatment of cancer TMSB10, PNMT, HNMT LOXL2 4402/4885CYP2D6 3599/4885HIF1A 692/4885
US-20170319535-A1 COMPOUNDS FOR USE IN THE PREVENTION OR TREATMENT OF CANCER TMSB10, PNMT, HNMT LOXL2 4454/4885CYP2D6 3495/4885HIF1A 646/4885
US-20260027148-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS SLC6A3, SIGMAR1, SLC6A4 LOXL2 4379/4885CYP2D6 29/4885HIF1A 4611/4885
US-20100324300-A1 PROCESS FOR PREPARING OPTICALLY ACTIVE AMINOPENTANE DERIVATIVE, INTERMEDIATE AND PROCESS FOR PREPARING INTERMEDIATE API5, CASP5, BAD LOXL2 3348/4885CYP2D6 232/4885HIF1A 3419/4885
US-20250345458-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS MC2R, SLC26A3, SLC5A1 LOXL2 3319/4885CYP2D6 1426/4885HIF1A 4577/4885
US-12472201-B2 Complexing agent salt formulations of pharmaceutical compounds SLC10A1, SLC5A6, MC2R LOXL2 3607/4885CYP2D6 1358/4885HIF1A 4621/4885
US-20260014190-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS SIGMAR1, OPRK1, SLC6A2 LOXL2 3606/4885CYP2D6 26/4885HIF1A 3731/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.