SCHEMBL2744582

SCHEMBL2744582

O=C(O)c1cn(C2CC2)c2ccc(F)cc2c1=O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.59
TOP2A P11388 6/20 0.57
TOP2B Q02880 6/20 0.57
ALDH1A1 P00352 4/20 0.57
LMNA P02545 3/20 0.57
HPGD P15428 2/20 0.57
HSD17B10 Q99714 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C9 P11712 1/20 0.57
MAPT P10636 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
PIK3CG P48736 4/20 0.48
PIK3CD O00329 3/20 0.48
PIK3R1 P27986 3/20 0.48
PIK3CA P42336 3/20 0.48
DPP4 P27487 1/20 0.47
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29766836 1.00 KDM4E (0.59) KDM4ETOP2ATOP2BALDH1A1LMNA
Hydrochloric Acid SCHEMBL6004997 0.99 KDM4E (0.57) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL28458144 0.99 KDM4E (0.57) KDM4ETOP2ATOP2BALDH1A1LMNA
Trifluoroacetic Acid SCHEMBL3808640 0.94 KDM4E (0.53) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL9146620 0.89 KDM4E (0.59) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL29518174 0.88 MEN1 (0.60) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL22506561 0.88 HTR3A (0.47) KDM4ETOP2ATOP2BALDH1A1LMNA
Potassium Ion SCHEMBL22497604 0.87 KDM4E (0.44) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL24616680 0.85 HTR3A (0.47) KDM4ETOP2ATOP2BALDH1A1LMNA
SCHEMBL6166633 0.84 KDM4E (0.48) KDM4ETOP2ATOP2BALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101068821-A Hybrid QA molecules where Q is an aminoquinoline and A is an antibiotic residue, their synthesis and use as antibacterial agents PALUMED SA (FR) 2007-11-07 CN claimed
EP-0169993-B1 7-(3-ARYL-1-PIPERAZINYL) AND 7-(3-CYCLOHEXYL-1-PIPERAZINYL) 3-QUINOLINE CARBOXYLIC ACIDS BAYER AG (DE) 1988-12-28 EP claimed
EP-0117474-A1 Quinolone carboxylic acids, process for their preparation and antibacterial compositions containing them BAYER AG (DE) 1984-09-05 EP claimed
EP-3929180-B1 QUINOLINE CARBOXYLIC ACID ESTER COMPOUND AND PREPARATION METHOD AND USE THEREOF SHANDONG UNITED PESTICIDE IND CO LTD (CN) 2026-03-04 EP disclosed
US-20250313533-A1 QUINOLINE CARBOXYLIC ACID ESTER COMPOUND AND PREPARATION METHOD AND USE THEREOF SHANDONG UNITED PESTICIDE INDUSTRY CO., LTD. (CN) 2025-10-09 US disclosed
US-11970487-B1 7-(4-((5-(benzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2h)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory and anticancer compound King Faisal University (SA) 2024-04-30 US disclosed
US-11873299-B1 7-(4-((5-(4-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)iperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound King Faisal University (SA) 2024-01-16 US disclosed
US-20220220076-A1 QUINOLINE CARBOXYLATE COMPOUND AND PREPARATION METHOD AND USE THEREOF SHANDONG UNITED PESTICIDE INDUSTRY CO., LTD. (CN) 2022-07-14 US disclosed
US-20220220076-A1 QUINOLINE CARBOXYLATE COMPOUND AND PREPARATION METHOD AND USE THEREOF SHANDONG UNITED PESTICIDE INDUSTRY CO., LTD. (CN) 2022-07-14 US disclosed
US-11261205-B2 Oxazolidinone-quinolone hybrid antibacterial for the parenteral treatment of prophylaxis of bacterial diseases MORPHOCHEM GMBH (DE) 2022-03-01 US disclosed
EP-3929180-A1 QUINOLINE CARBOXYLIC ACID ESTER COMPOUND AND PREPARATION METHOD AND USE THEREOF Shandong United Pesticide Industry Co., Ltd. (CN) 2021-12-29 EP disclosed
EP-0641793-A1 5-Amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative HOKURIKU SEIYAKU CO., LTD. (JP) 1995-03-08 EP disclosed
US-5300644-A Process for the preparation of quinoline carboxylic acids CHINOIN GYOGYSER- ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1994-04-05 US disclosed
CN-1074218-A Quinolone-and naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1993-07-14 CN disclosed
EP-0237955-B1 QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR PREPARATION KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-07-15 EP disclosed
US-5091530-A BARON CHELATES OF QUINOLINE CARBOXYLIC ACIDS CHINOIN GYOGYSZER- ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1992-02-25 US disclosed
CN-88101907-A Process for preparing quinoline carboxylic acids 1988-10-26 CN disclosed
CN-85101832-A The method for preparing 7-(3-aryl-1-piperazinyl)-3-quinolone carboxylic acid and 7-(3-encircles ethyl-1-piperazinyl)-3-quinolone carboxylic acid 1987-01-31 CN disclosed
EP-0113092-B1 1-CYCLOPROPYL-6-FLUORO-1,4-DIHYDRO-4-OXO-7-(4-(OXOALKYL)-1-PIPERAZINYL)-3-QUINOLINE-CARBOXYLIC ACIDS AND THEIR DERIVATIVES, PROCESS FOR THEIR PREPARATION AND ANTIBACTERIAL AGENTS CONTAINING THEM BAYER AG (DE) 1986-05-21 EP disclosed
EP-0117474-A1 Quinolone carboxylic acids, process for their preparation and antibacterial compositions containing them BAYER AG (DE) 1984-09-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250313533-A1 QUINOLINE CARBOXYLIC ACID ESTER COMPOUND AND PREPARATION METHOD AND USE THEREOF NAAA, SDHA, GLUL KDM4E 858/4885TOP2A 681/4885TOP2B 930/4885
US-11873299-B1 7-(4-((5-(4-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)iperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound DPP4, IL1A, IL1B KDM4E 881/4885TOP2A 255/4885TOP2B 553/4885
US-11970487-B1 7-(4-((5-(benzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2h)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory and anticancer compound IL1A, NFKBIA, CASP1 KDM4E 1046/4885TOP2A 34/4885TOP2B 68/4885
US-11261205-B2 Oxazolidinone-quinolone hybrid antibacterial for the parenteral treatment of prophylaxis of bacterial diseases NQO2, QARS1, RECQL KDM4E 4487/4885TOP2A 56/4885TOP2B 85/4885
US-20220220076-A1 QUINOLINE CARBOXYLATE COMPOUND AND PREPARATION METHOD AND USE THEREOF SDHA, GLUL, PGLS KDM4E 1227/4885TOP2A 169/4885TOP2B 280/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.