SCHEMBL275643

SCHEMBL275643

O=S(=O)(O)c1cc(S(=O)(=O)O)c2nc(-c3ccc(-c4nc5c(S(=O)(=O)O)cccc5[nH]4)cc3)[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.49
DHODH Q02127 7/20 0.47
PARP1 P09874 9/20 0.46
MGAM O43451 3/20 0.43
GAA P10253 3/20 0.43
SI P14410 3/20 0.43
MGAM2 Q2M2H8 3/20 0.43
HPSE Q9Y251 1/20 0.41
PARP2 Q9UGN5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bisdisulizole SCHEMBL29507075 0.92 HDAC6 (0.52) HDAC6DHODHPARP1GAA
Bisdisulizole SCHEMBL62139 0.92 HDAC6 (0.52) HDAC6DHODHPARP1GAA
Bisdisulizole SCHEMBL29507102 0.92 HDAC6 (0.52) HDAC6DHODHPARP1GAA
Bisdisulizole SCHEMBL1830829 0.91 HDAC6 (0.51) HDAC6DHODHPARP1GAA
Bisdisulizole SCHEMBL4777834 0.91 HDAC6 (0.51) HDAC6DHODHPARP1GAA
SCHEMBL6575742 0.88 HDAC6 (0.63) HDAC6DHODHPARP1GAA
SCHEMBL14224890 0.85 HDAC6 (0.46) HDAC6DHODHPARP1GAA
SCHEMBL22902385 0.85 HDAC6 (0.46) HDAC6DHODHPARP1GAA
SCHEMBL20848229 0.85 HDAC6 (0.46) HDAC6DHODHMGAMGAASI
Bisdisulizole SCHEMBL1830834 0.85 HDAC6 (0.49) HDAC6DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210346249-A1 COMPOSITION COMPRISING A UV-SCREENING AGENT, AN ANIONIC CROSSLINKED HYDROPHILIC POLYMER, A SURFACTANT HAVING AN HLB LESS THAN OR EQUAL TO 5 AND A SILICONE COPOLYMER L'OREAL (FR) 2021-11-11 US disclosed
EP-3185843-B1 GEL COMPOSITION AND GEL COMPRISING A UV FILTER OREAL (FR) 2021-08-11 EP disclosed
EP-3389618-B1 PROCESS FOR TREATING KERATIN FIBRES USING AN AQUEOUS COMPOSITION COMPRISING A COMBINATION OF PARTICULAR ALKOXYSILANES OREAL (FR) 2021-01-20 EP disclosed
EP-3389604-B1 COMPOSITION COMPRISING A COMBINATION OF PARTICULAR ALKOXYSILANES AND A FATTY SUBSTANCE OREAL (FR) 2020-04-08 EP disclosed
US-20200030200-A1 COMPOSITION COMPRISING A UV-SCREENING AGENT, AN ANIONIC CROSSLINKED HYDROPHILIC POLYMER, A SURFACTANT HAVING AN HLB LESS THAN OR EQUAL TO 5 AND A SILICONE COPOLYMER L'OREAL (FR) 2020-01-30 US disclosed
EP-3307233-B1 COMPOSITION COMPRISING A UV-SCREENING AGENT, AN ANIONIC CROSSLINKED HYDROPHILIC POLYMER, A SURFACTANT HAVING AN HLB LESS THAN OR EQUAL TO 5 AND A SILICONE COPOLYMER OREAL (FR) 2019-11-06 EP disclosed
EP-2945603-B1 COSMETIC OR DERMATOLOGICAL COMPOSITION COMPRISING A MEROCYANINE AND A UVA-SCREENING AGENT OF THE AMINO-SUBSTITUTED 2-HYDROXYBENZOPHENONE TYPE AND/OR A HYDROPHILIC ORGANIC UVA-SCREENING AGENT OREAL (FR) 2019-03-27 EP disclosed
WO-2019002494-A1 USE OF A WASHING COMPOSITION COMPRISING SURFACTANTS AND CATIONIC AND/OR AMPHOTERIC POLYMERS IN COMBINATION WITH A COMPOSITION COMPRISING ANIONIC BENEFICIAL AGENTS L'OREAL (FR) 2019-01-03 WO disclosed
US-9926289-B2 Compositions, apparatus, systems, and methods for resolving electronic excited states BANK OF AMERICA, N.A., AS ADMINISTRATIVE AGENT 2018-03-27 US disclosed
US-20170326045-A1 COSMETIC COMPOSITION COMPRISING A SYNTHETIC PHYLLOSILICATE AND A POLYOL AND/OR A UV FILTER L'OREAL (FR) 2017-11-16 US disclosed
US-8278332-B2 Photostabilization of retinoids with alkoxycrylene compounds HALLSTAR INNOVATIONS CORP. (US) 2012-10-02 US disclosed
US-8268294-B2 Photostabilization of retinoids with alkoxycrylene compounds HALLSTAR INNOVATIONS CORP. (US) 2012-09-18 US disclosed
US-8263051-B2 Photostabilization of resveratrol with alkoxycrylene compounds HALLSTAR INNOVATIONS CORP. (US) 2012-09-11 US disclosed
US-20120148512-A1 Method for Increasing the Sun Protection Factor of a Cosmetic and/or Dermatological Preparation BASF SE (DE) 2012-06-14 US disclosed
US-20120065232-A1 PHOTOSTABILIZATION OF RETINOIDS WITH ALKOXYCRYLENE COMPOUNDS HALLSTAR INNOVATIONS CORP. (US) 2012-03-15 US disclosed
US-8133477-B2 Dispersions of inorganic particulates containing alkoxycrylene HALLSTAR INNOVATIONS CORP. (US) 2012-03-13 US disclosed
US-20110268674-A1 POLYAMIDE-5 COMPOUNDS IN COSMETIC PREPARATIONS BEIERSDORF AG (DE) 2011-11-03 US disclosed
US-20110251242-A1 PHOTOSTABILIZATION OF RESVERATROL WITH ALKOXYCRYLENE COMPOUNDS HALLSTAR INNOVATIONS CORP. (US) 2011-10-13 US disclosed
US-20110142771-A1 Photostabilization of Retinoids with Alkoxycrylene Compounds HALLSTAR INNOVATIONS CORP. (US) 2011-06-16 US disclosed
US-20100021403-A1 DISPERSIONS OF INORGANIC PARTICULATES CONTAINING ALKOXYCRYLENE HALLSTAR INNOVATIONS CORP. (US) 2010-01-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100021403-A1 DISPERSIONS OF INORGANIC PARTICULATES CONTAINING ALKOXYCRYLENE C9, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, SIGMAR1 HDAC6 3261/4885DHODH 4517/4885PARP1 1087/4885
US-20120148512-A1 Method for Increasing the Sun Protection Factor of a Cosmetic and/or Dermatological Preparation CUTA, ERCC4, SUN2 HDAC6 2296/4885DHODH 536/4885PARP1 2331/4885
US-20110268674-A1 POLYAMIDE-5 COMPOUNDS IN COSMETIC PREPARATIONS CUTA, PLIN5, PGA5 HDAC6 344/4885DHODH 4129/4885PARP1 268/4885
US-20110142771-A1 Photostabilization of Retinoids with Alkoxycrylene Compounds RBP4, RARA, RBP1 HDAC6 4824/4885DHODH 1525/4885PARP1 1551/4885
US-20170326045-A1 COSMETIC COMPOSITION COMPRISING A SYNTHETIC PHYLLOSILICATE AND A POLYOL AND/OR A UV FILTER PUF60, POLR1C, DPM1 HDAC6 2024/4885DHODH 3751/4885PARP1 1633/4885
US-20200030200-A1 COMPOSITION COMPRISING A UV-SCREENING AGENT, AN ANIONIC CROSSLINKED HYDROPHILIC POLYMER, A SURFACTANT HAVING AN HLB LESS THAN OR EQUAL TO 5 AND A SILICONE COPOLYMER ERCC5, CUTA, PLIN5 HDAC6 4356/4885DHODH 1364/4885PARP1 2740/4885
US-20120065232-A1 PHOTOSTABILIZATION OF RETINOIDS WITH ALKOXYCRYLENE COMPOUNDS RBP4, RARA, RBP1 HDAC6 4823/4885DHODH 1620/4885PARP1 1510/4885
US-20210346249-A1 COMPOSITION COMPRISING A UV-SCREENING AGENT, AN ANIONIC CROSSLINKED HYDROPHILIC POLYMER, A SURFACTANT HAVING AN HLB LESS THAN OR EQUAL TO 5 AND A SILICONE COPOLYMER ERCC5, CUTA, PLIN5 HDAC6 4356/4885DHODH 1364/4885PARP1 2740/4885
US-20110251242-A1 PHOTOSTABILIZATION OF RESVERATROL WITH ALKOXYCRYLENE COMPOUNDS CBR1, CBR3, PC HDAC6 4476/4885DHODH 1973/4885PARP1 251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.