Glybuthiazol

Glybuthiazol

SCHEMBL282607

CC(C)(C)c1nnc(NS(=O)(=O)c2ccc(N)cc2)s1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.71
HPGD P15428 2/20 0.71
HSD17B10 Q99714 2/20 0.71
MAPT P10636 2/20 0.71
TSHR P16473 1/20 0.71
LMNA P02545 1/20 0.68
PKM P14618 1/20 0.67
AKT1 P31749 4/20 0.63
CA1 P00915 3/20 0.62
CA2 P00918 3/20 0.62
CA5A P35218 2/20 0.62
CA5B Q9Y2D0 2/20 0.62
CA12 O43570 1/20 0.62
CA3 P07451 1/20 0.62
CA6 P23280 1/20 0.62
CA9 Q16790 1/20 0.62
CA14 Q9ULX7 1/20 0.62
CA4 P22748 1/20 0.59
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30978753 0.86 MEN1 (0.75) ALDH1A1HPGDHSD17B10MAPTTSHR
SCHEMBL5404442 0.86 ALDH1A1 (0.71) ALDH1A1HPGDHSD17B10MAPTTSHR
Glybuzole SCHEMBL34401 0.85 ALDH1A1 (0.71) ALDH1A1HPGDHSD17B10MAPTTSHR
SCHEMBL30578971 0.83 ALDH1A1 (1.00) ALDH1A1HPGDHSD17B10MAPTTSHR
Sulfamethizole SCHEMBL26453 0.81 ALDH1A1 (1.00) ALDH1A1HPGDLMNAPKMAKT1
SCHEMBL286763 0.80 ALDH1A1 (1.00) ALDH1A1HPGDHSD17B10MAPTTSHR
Sulfamethizole SCHEMBL1566142 0.79 ALDH1A1 (0.97) ALDH1A1HPGDLMNAPKMAKT1
SCHEMBL5401782 0.79 ALDH1A1 (0.65) ALDH1A1HPGDHSD17B10MAPTTSHR
Sulfamethizole SCHEMBL28693374 0.78 ALDH1A1 (0.94) ALDH1A1HPGDLMNAPKMAKT1
SCHEMBL328580 0.78 LMNA (0.68) ALDH1A1TSHRLMNAAKT1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1470 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021054927-A2 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2021-03-25 WO claimed
EP-2459227-B1 Prodrugs containing an aromatic amine connected by an amide bond to a carrier ASCENDIS PHARMA AS (DK) 2021-03-17 EP claimed
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2020-02-13 US claimed
US-9622969-B2 Polymer conjugated protein micelles SOUTH DAKOTA STATE UNIV (US) 2017-04-18 US claimed
US-9173953-B2 Prodrugs containing an aromatic amine connected by an amido bond to a linker ASCENDIS PHARMA AS (DK) 2015-11-03 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20140370110-A1 POLYMER CONJUGATED PROTEIN MICELLES SOUTH DAKOTA STATE UNIVERSITY (US) 2014-12-18 US claimed
US-20140296141-A1 Compositions and Methods for Treating Obesity, Obesity Related Disorders and for Inhibiting the Infectivity of Human Immunodeficiency Virus THE GENERAL HOSPITAL CORPORATION (US) 2014-10-02 US claimed
US-8591947-B2 Dual controlled release dosage form Osmotica Kereskedelmi és Szolgáltató KFT (HU) 2013-11-26 US claimed
US-20130108693-A1 Dual Controlled Release Dosage Form OSMOTICA KERESKEDELMI ES SZOLGALTATO KFT (HU) 2013-05-02 US claimed
WO-2002015892-A2 COMBINATION COMPRISING AN INSULIN SECRETION ENHANCER AND AN ACTIVE INGREDIENT SELECTED FROM HMG-CO-A REDUCTASE INHIBITORS AND ACE INHIBITORS NOVARTIS AG (CH) 2002-02-28 WO claimed
WO-2002015933-A2 COMBINATION COMPRISING AN AT1-RECEPTOR ANTAGONIST AND AN INSULIN SECRETION ENHANCER OR AN INSULIN SENSITISER NOVARTIS AG (CH) 2002-02-28 WO claimed
US-6329404-B1 Pharmaceutical composition TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-11 US claimed
US-6303640-B1 ADMINISTERING OXAZOLE OR THIAZOLE DERIVATIVE COMPOUND FOR REDUCING SIDE EFFECTS OF DIABETIC THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-10-16 US claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
US-6211205-B1 ANTIDIABETIC AGENTS THAT ENHANCE INSULIN SECRETION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US claimed
US-6150383-A COMPRISING AN INSULIN SENSITIVITY ENHANCER IN COMBINATION WITH ONE OR MORE OTHER ANTIDIABETICS DIFFERING FROM THE ENHANCER IN MECHANISM OF ACTION; LIPID/GLYCOMETABOLISM DISORDERS; ANTIDIABETIC AGENTS; SIDE EFFECT REDUCTION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-11-21 US claimed
EP-0007911-A4 ZINC AND/OR CERIUM CONTAINING SULFONYLUREA HYPOGLYCEMIC AGENTS, PREPARATION AND USE THEREOF. RESEARCH CORP (US) 1981-02-25 EP claimed
EP-0007911-A1 ZINC AND/OR CERIUM CONTAINING SULFONYLUREA HYPOGLYCEMIC AGENTS, PREPARATION AND USE THEREOF Research Corporation (US) 1980-02-06 EP claimed
WO-1979000435-A1 ZINC AND/OR CERIUM CONTAINING SULFONYLUREA HYPOGLYCEMIC AGENTS,PREPARATION AND USE THEREOF RESEARCH CORP (US) 1979-07-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS GSTK1, GSTO1, GSTM2 ALDH1A1 2491/4885HPGD 348/4885HSD17B10 492/4885
US-20140370110-A1 POLYMER CONJUGATED PROTEIN MICELLES MTDH, PSMG3, GHITM ALDH1A1 4150/4885HPGD 2962/4885HSD17B10 3318/4885
US-20140296141-A1 Compositions and Methods for Treating Obesity, Obesity Related Disorders and for Inhibiting the Infectivity of Human Immunodeficiency Virus LPL, ADIPOR2, EBP ALDH1A1 884/4885HPGD 1103/4885HSD17B10 50/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.