SCHEMBL28296378

SCHEMBL28296378

N#Cc1cc(N(C(=O)c2ccccc2)S(=O)(=O)c2ccccc2)ccc1N1CCN(CCOC=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.38
DRD4 P21917 5/20 0.38
HSP90AA1 P07900 1/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
GMNN O75496 1/20 0.35
THRB P10828 1/20 0.35
PMP22 Q01453 1/20 0.35
KCNA5 P22460 1/20 0.35
DRD3 P35462 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTR2A P28223 1/20 0.35
THPO P40225 1/20 0.35
HIF1A Q16665 1/20 0.35
GAA P10253 2/20 0.34
HTR7 P34969 2/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethoxycarbonyl Group SCHEMBL28296379 0.83 HTR6 (0.37) HSP90AA1ALDH1A1KDM4ELMNADRD3
SCHEMBL28294727 0.83 NR3C1 (0.42) ALDH1A1LMNADRD3HTR2AGAA
SCHEMBL28744897 0.80 MAPK1 (0.49) ALDH1A1KDM4ELMNAGAAMAPT
SCHEMBL28294730 0.76 ALDH1A1 (0.53) DRD2DRD4ALDH1A1KDM4ELMNA
SCHEMBL28873296 0.71 MAPT (0.50) DRD2ALDH1A1KDM4ELMNADRD3
SCHEMBL28296408 0.70 LTA4H (0.43) DRD2DRD4ALDH1A1KDM4ELMNA
SCHEMBL28296376 0.65 NR3C1 (0.47) ALDH1A1LMNADRD3HTR2AHTR7
SCHEMBL28294734 0.65 LMNA (0.41) DRD4ALDH1A1KDM4ELMNADRD3
SCHEMBL28744878 0.64 USP2 (0.55) ALDH1A1KDM4ELMNAGAAKMT2A
SCHEMBL28744845 0.64 MAPK1 (0.54) ALDH1A1LMNAGAAMAPTRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651297-A A kind of N- benzyl-N- aryl sulfonic acid amides analog derivative and preparation and application 杭州壹瑞医药科技有限公司 2019-04-19 CN claimed
CN-109651297-A A kind of N- benzyl-N- aryl sulfonic acid amides analog derivative and preparation and application 杭州壹瑞医药科技有限公司 2019-04-19 CN disclosed