SCHEMBL28296408

SCHEMBL28296408

N#Cc1cc(NCc2ccccc2)ccc1N1CCN(CCOC=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.43
HTR6 P50406 4/20 0.42
GAA P10253 3/20 0.42
HTR2A P28223 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
DRD2 P14416 5/20 0.41
HTR1A P08908 4/20 0.41
HTR7 P34969 3/20 0.41
LMNA P02545 1/20 0.39
ACHE P22303 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28957487 0.90 GAA (0.43) HTR6GAAALDH1A1HPGDKDM4E
SCHEMBL28294734 0.83 LMNA (0.41) GAAHTR2AALDH1A1HPGDKDM4E
SCHEMBL28294730 0.82 ALDH1A1 (0.53) HTR2AALDH1A1HPGDKDM4EDRD2
Ethoxycarbonyl Group SCHEMBL28296409 0.80 ALDH1A1 (0.41) HTR6GAAHTR2AALDH1A1HPGD
SCHEMBL28873296 0.77 MAPT (0.50) GAAHTR2AALDH1A1KDM4EDRD2
SCHEMBL28294727 0.75 NR3C1 (0.42) HTR6GAAHTR2AALDH1A1HPGD
Ethoxycarbonyl Group SCHEMBL28957488 0.71 GAA (0.42) HTR6GAAALDH1A1HPGDKDM4E
SCHEMBL28296378 0.70 DRD2 (0.38) HTR6GAAHTR2AALDH1A1KDM4E
SCHEMBL22273612 0.70 KDM4E (0.42) HTR6GAAHTR2AALDH1A1HPGD
SCHEMBL7262207 0.69 KCNH2 (0.57) HTR2ADRD2HTR1AHTR7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651297-A A kind of N- benzyl-N- aryl sulfonic acid amides analog derivative and preparation and application 杭州壹瑞医药科技有限公司 2019-04-19 CN disclosed