SCHEMBL28822841

SCHEMBL28822841

Cc1ccc(-c2sc(C=O)c(-c3ccc(CN)cc3)c2N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 2/20 0.34
LTA4H P09960 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
XBP1 P17861 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NEK1 Q96PY6 1/20 0.34
F9 P00740 1/20 0.33
F11 P03951 1/20 0.33
F7 P08709 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
RAB9A P51151 1/20 0.32
DUSP3 P51452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27975865 0.88 TAAR1 (0.46) HRH3LMNALTA4HKDM4EMAPT
SCHEMBL28036394 0.85 ALOX5 (0.39) SMN1; SMN2LMNAKDM4EMAPTXBP1
SCHEMBL28036416 0.83 PTGS2 (0.47) SMN1; SMN2LMNAKDM4EMAPTXBP1
SCHEMBL28822843 0.82 HTR7 (0.35) HRH3LTA4HNEK1NOS3NOS1
SCHEMBL27975845 0.82 LOXL2 (0.51) SMN1; SMN2LMNAMAPTMAPK1NPSR1
SCHEMBL28036417 0.79 ACHE (0.46) SMN1; SMN2LMNAMAPTMAPK1NPSR1
SCHEMBL27975859 0.75 ALDH1A1 (0.37) SMN1; SMN2LMNAKDM4EMAPTCYP2C9
SCHEMBL28036701 0.74 SIRT1 (0.40) LMNAKDM4EMAPTNPSR1ALDH1A1
SCHEMBL27975546 0.70 ALDH1A1 (0.40) SMN1; SMN2LMNAKDM4EMAPTMAPK1
SCHEMBL27975579 0.70 TP53 (0.43) MAPTMAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980248-B 3,5-bis-substituted-4-amino thiophene-2-formaldehyde compound and preparation method thereof ZHEJIANG UNIVERSITY (CN) 2015-11-18 CN disclosed