SCHEMBL289310

SCHEMBL289310

FC(F)(F)c1cccc(OBOc2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAOB P27338 1/20 0.44
AOC3 Q16853 1/20 0.44
PPARG P37231 4/20 0.43
IDO1 P14902 2/20 0.43
PPARA Q07869 1/20 0.43
CES2 O00748 1/20 0.42
MGLL Q99685 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6113954 0.84 MAOB (0.40) TSHRMAPK1L3MBTL1SLC6A2SLC6A4
SCHEMBL121487 0.84 KDM4E (0.46) TSHRMAPK1L3MBTL1SLC6A2SLC6A4
SCHEMBL9798371 0.80 LTA4H (0.54) TSHRMAPK1L3MBTL1SLC6A2SLC6A4
SCHEMBL841548 0.79 CYP3A4 (0.46) MAPK1L3MBTL1PPARGLMNAHSD17B10
SCHEMBL4506704 0.78 PPARG (0.40) KDM4EMAOBPPARGPPARACES2
SCHEMBL521971 0.78 IDO1 (0.40) TSHRIDO1CES2ALDH1A1
SCHEMBL5608697 0.77 TSHR (0.48) TSHRMAPK1L3MBTL1SLC6A2SLC6A4
SCHEMBL4214531 0.77 TSHR (0.54) TSHRMAPK1L3MBTL1SLC6A2SLC6A4
SCHEMBL167016 0.77 L3MBTL1 (0.58) TSHRMAPK1L3MBTL1KDM4EMAOB
SCHEMBL11527555 0.77 KIF11 (0.51) TSHRMAPK1L3MBTL1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 473 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105732574-A Preparation of thianthrene-5, 5,10, 10-tetraoxide derivative and organic electroluminescent device based on thianthrene-5, 5,10, 10-tetraoxide derivative 中国科学院理化技术研究所 2016-07-06 CN claimed
CN-105693608-A 2, 2-dimethyl-1, 3-indene dione derivatives and organic electroluminescent devices based thereon 中国科学院理化技术研究所 2016-06-22 CN claimed
CN-105220473-A A kind of water-proof aagent and application thereof HOPERISE TEXTILES CO LTD QUANZHOU 2016-01-06 CN claimed
US-20250388582-A1 NOVEL BICYCLIC HETEROARYL COMPOUND AND USE THEREOF ILDONG PHARMACEUTICAL CO LTD (KR) 2025-12-25 US disclosed
US-20250333383-A1 N-OXIDE COMPOUNDS AND USE THEREOF SK BIOPHARMACEUTICALS CO., LTD. (KR) 2025-10-30 US disclosed
US-20250282735-A1 BICYCLE COMPOUNDS AS TEAD INHIBITOR DONG-A ST CO., LTD. (KR) 2025-09-11 US disclosed
US-20250214969-A1 PROTEIN DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-07-03 US disclosed
US-20250179017-A1 CARBOXAMIDE COMPOUNDS AS PGE2 RECEPTOR ANTAGONISTS GUANGDONG NEWOPP BIOPHARMACEUTICALS CO., LTD. (CN) 2025-06-05 US disclosed
WO-2025110621-A1 NOVEL OXAZOLE-BASED COMPOUND AND COMPOSITION FOR PREVENTING, ALLEVIATING, OR TREATING INFLAMMATORY DISEASES COMPRISING SAME 고려대학교 세종산학협력단 2025-05-30 WO disclosed
US-12312337-B2 Compounds and methods for treating cancer ANTIDOTE IP HOLDINGS, LLC (US) 2025-05-27 US disclosed
CN-119874668-A Main protease regulator and application thereof 北京昌平实验室 2025-04-25 CN disclosed
EP-1077929-A1 2,3,5-SUBSTITUTED BIPHENYLS USEFUL IN THE TREATMENT OF INSULIN RESISTANCE AND HYPERGLYCEMIA AMERICAN HOME PRODUCTS CORPORATION (US) 2001-02-28 EP disclosed
WO-2000046184-A1 N2-PHENYLAMIDINE DERIVATIVES AVENTIS CROPSCIENCE GMBH (FR) 2000-08-10 WO disclosed
WO-1999061410-A1 2,3,5-SUBSTITUTED BIPHENYLS USEFUL IN THE TREATMENT OF INSULIN RESISTANCE AND HYPERGLYCEMIA AMERICAN HOME PRODUCTS CORPORATION (US) 1999-12-02 WO disclosed
EP-0691966-B1 QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS SYNTEX INC (US) 1998-09-09 EP disclosed
US-5530005-A THERAPY FOR SKIN DISORDERS, AIDS, IMMUNOSUPPRESION DISEASES SYNTEX (U.S.A.) INC. (US) 1996-06-25 US disclosed
EP-0691966-A1 QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1996-01-17 EP disclosed
US-5475003-A Antiinflammatory agent, immunosuppressive, antiallergens, bronchodilators, analgens SYNTEX (U.S.A.) INC. (US) 1995-12-12 US disclosed
US-5455252-A Antiinflammatory agent, immunosuppressant, antiallergen, skin disorders, bronchodilator, analgesic SYNTEX (U.S.A.) INC. (US) 1995-10-03 US disclosed
WO-1994022852-A1 QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1994-10-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179017-A1 CARBOXAMIDE COMPOUNDS AS PGE2 RECEPTOR ANTAGONISTS PTGER1, PTGER2, CNR2 TSHR 489/4885MAPK1 1164/4885L3MBTL1 4743/4885
US-20250333383-A1 N-OXIDE COMPOUNDS AND USE THEREOF SCNN1B, SCN1B, SCN2B TSHR 2806/4885MAPK1 1015/4885L3MBTL1 4726/4885
US-20250282735-A1 BICYCLE COMPOUNDS AS TEAD INHIBITOR TEAD1, TEAD2, TEAD3 TSHR 3560/4885MAPK1 1623/4885L3MBTL1 4484/4885
US-20250214969-A1 PROTEIN DEGRADERS AND USES THEREOF MDM2, CUL1, PSMG3 TSHR 3432/4885MAPK1 3746/4885L3MBTL1 969/4885
US-20250388582-A1 NOVEL BICYCLIC HETEROARYL COMPOUND AND USE THEREOF GBA1, PIKFYVE, MAN2B1 TSHR 3647/4885MAPK1 1105/4885L3MBTL1 816/4885
US-12312337-B2 Compounds and methods for treating cancer AHR, ARNT, HMOX1 TSHR 2669/4885MAPK1 2405/4885L3MBTL1 3525/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.