SCHEMBL2913743

SCHEMBL2913743

[C-]#[N+]c1cccc([N+](=O)[O-])c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.61
LMNA P02545 2/20 0.61
ALDH1A1 P00352 6/20 0.52
ACHE P22303 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALOX15 P16050 1/20 0.52
HSP90AA1 P07900 1/20 0.50
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
KMT2A Q03164 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
TP53 P04637 1/20 0.47
NFE2L2 Q16236 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46
FBP1 P09467 1/20 0.44
VCP P55072 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11290393 0.98 TSHR (0.59) TSHRLMNAALDH1A1ACHETDP1
Hydrochloric Acid SCHEMBL11290386 0.98 TSHR (0.59) TSHRLMNAALDH1A1ACHETDP1
SCHEMBL28239092 0.80 TSHR (0.61) TSHRLMNAALDH1A1ACHETDP1
Hydrochloric Acid SCHEMBL11567135 0.78 TSHR (0.59) TSHRLMNAALDH1A1ACHETDP1
Dinitrophenylene SCHEMBL36632 0.78 TSHR (1.00) TSHRLMNAALDH1A1ACHETDP1
Dinitrophenylene SCHEMBL29291896 0.78 TSHR (1.00) TSHRLMNAALDH1A1ACHETDP1
Perchlorate SCHEMBL5574429 0.76 TSHR (0.55) TSHRLMNAALDH1A1ACHETDP1
Dinitrophenylene SCHEMBL9733868 0.75 TSHR (0.94) TSHRLMNAALDH1A1ACHETDP1
Dinitrophenylene SCHEMBL11661349 0.75 TSHR (0.94) TSHRLMNAALDH1A1ACHETDP1
Dinitrophenylene SCHEMBL2997371 0.75 TSHR (0.94) TSHRLMNAALDH1A1ACHETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11655203-B2 Nitration ETH ZURICH (CH) 2023-05-23 US disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-20180057465-A1 Inhibitors of Necroptosis CATALYST THERAPEUTICS PTY LTD (AU) 2018-03-01 US disclosed
US-20170247352-A1 METHOD FOR PREPARING ALECTINIB SUZHOU MIRACPHARMA TECHNOLOGY CO., LTD. (CN) 2017-08-31 US disclosed
US-9573932-B2 Synthesis of intermediates in the preparation of ALK inhibitor XU YONG (US) 2017-02-21 US disclosed
US-20160257667-A1 SYNTHESIS OF INTERMEDIATES IN THE PREPARATION OF ALK INHIBITOR XU YONG (US) 2016-09-08 US disclosed
US-20150038534-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. 2015-02-05 US disclosed
US-8901156-B2 Compounds and methods TEMPERO PHARMACEUTICALS, INC. (US) 2014-12-02 US disclosed
US-20130059883-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. 2013-03-07 US disclosed
EP-1901748-B1 ANGIOGENESIS INHIBITORS ONCALIS AG (CH) 2010-09-08 EP disclosed
EP-1765351-B9 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2010-03-24 EP disclosed
EP-1765351-B1 PROTEIN KINASE INHIBITORS ONCALIS AG (CH) 2009-03-04 EP disclosed
WO-2008121602-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160257667-A1 SYNTHESIS OF INTERMEDIATES IN THE PREPARATION OF ALK INHIBITOR ALK, ACVR1B, ETV6 TSHR 3480/4885LMNA 1093/4885ALDH1A1 439/4885
US-20150038534-A1 COMPOUNDS AND METHODS XDH, LPXN, CCNY TSHR 1016/4885LMNA 26/4885ALDH1A1 1152/4885
US-20170247352-A1 METHOD FOR PREPARING ALECTINIB ADH1C, ADH1A, ALK TSHR 2007/4885LMNA 376/4885ALDH1A1 166/4885
US-20130059883-A1 COMPOUNDS AND METHODS XDH, LPXN, CCNY TSHR 1016/4885LMNA 26/4885ALDH1A1 1152/4885
US-20180057465-A1 Inhibitors of Necroptosis RIPK3, RIPK1, AIFM1 TSHR 4108/4885LMNA 1012/4885ALDH1A1 4651/4885
US-11655203-B2 Nitration NOS1, NOS2, NOS3 TSHR 2432/4885LMNA 4595/4885ALDH1A1 2335/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.