Flerobuterol

Flerobuterol

SCHEMBL29356232

CC(C)(C)NCC(O)c1ccccc1F

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.66
ADRB2 P07550 4/20 0.66
HIF1A Q16665 2/20 0.66
CYP2D6 P10635 2/20 0.66
NFKB1 P19838 1/20 0.66
BLM P54132 1/20 0.64
ADRB3 P13945 2/20 0.49
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
CASP7 P55210 1/20 0.45
KMT2A Q03164 1/20 0.45
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flerobuterol SCHEMBL249507 1.00 ADRB1 (0.66) ADRB1ADRB2HIF1ACYP2D6NFKB1
Flerobuterol SCHEMBL20819557 1.00 ADRB1 (0.66) ADRB1ADRB2HIF1ACYP2D6NFKB1
Flerobuterol SCHEMBL30956705 1.00 ADRB1 (0.66) ADRB1ADRB2HIF1ACYP2D6NFKB1
Flerobuterol SCHEMBL10624514 0.98 BLM (0.67) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL30956709 0.87 ADRB1 (0.58) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL20819687 0.87 ADRB1 (0.58) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL30956714 0.87 ADRB1 (0.58) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL9820962 0.87 ADRB1 (0.58) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL20819586 0.85 ADRB2 (0.56) ADRB1ADRB2HIF1ACYP2D6NFKB1
SCHEMBL20819585 0.85 ADRB2 (0.56) ADRB1ADRB2HIF1ACYP2D6NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116857-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOFS PARDES BIOSCIENCES INC (US) 2026-04-30 US disclosed
US-20250313573-A1 HYDROXYPYRIDOXAZEPINES AS NRF2 ACTIVATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2025-10-09 US disclosed
EP-4605396-A1 ANTICORONVIRAL COMPOUNDS AND COMPOSITIONS AND USES THEREOF Shanghai Curegene Pharmaceutical Co., Ltd. (CN) 2025-08-27 EP disclosed
WO-2025119207-A1 ANTIVIRAL COMPOUNDS AND COMPOSITIONS AND USES THEREOF SHANGHAI CUREGENE PHARMACEUTICAL CO., LTD. (CN) 2025-06-12 WO disclosed
EP-4252755-B1 THERAPEUTIC COMPOUNDS C4X DISCOVERY LTD (GB) 2025-05-14 EP disclosed
EP-4139295-B1 ISOQUINILINE NRF2 AGONISTS C4X DISCOVERY LTD (GB) 2025-04-09 EP disclosed
EP-4139294-B1 ISOQUINILINE NRF2 AGONISTS C4X DISCOVERY LTD (GB) 2025-04-09 EP disclosed
US-20250084075-A1 THERAPEUTIC COMPOUNDS C4X DISCOVERY LIMITED (GB) 2025-03-13 US disclosed
US-20250084077-A1 ETHER LINKED TRIAZOLES AS NRF2 ACTIVATORS ASTEX THERAPEUTICS LIMITED (GB) 2025-03-13 US disclosed
WO-2025011656-A1 ANTICORONVIRAL COMPOUNDS AND COMPOSITIONS AND USES THEREOF SHANGHAI CUREGENE PHARMACEUTICAL CO., LTD. (CN) 2025-01-16 WO disclosed
WO-2022221686-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2022-10-20 WO disclosed
US-11472793-B2 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2022-10-18 US disclosed
US-20220324875-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-10-13 US disclosed
US-20220324844-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2022-10-13 US disclosed
US-20220204526-A1 HYDROXYPYRIDOXAZEPINES AS NRF2 ACTIVATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-06-30 US disclosed
US-20220162194-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2022-05-26 US disclosed
US-11312704-B2 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2022-04-26 US disclosed
US-20220089590-A1 ETHER LINKED TRIAZOLES AS NRF2 ACTIVATORS ASTEX THERAPEUTICS LIMITED (GB) 2022-03-24 US disclosed
US-11260049-B2 TRPV4 antagonists GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2022-03-01 US disclosed
US-11229623-B2 TRPV4 antagonists GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2022-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11260049-B2 TRPV4 antagonists TRPV4, TRPV5, TRPV2 ADRB1 1180/4885ADRB2 1126/4885HIF1A 1995/4885
US-20220089590-A1 ETHER LINKED TRIAZOLES AS NRF2 ACTIVATORS NFE2L2, KEAP1, NQO1 ADRB1 871/4885ADRB2 965/4885HIF1A 439/4885
US-20260116857-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOFS CTRC, CTRL, CTSL ADRB1 4764/4885ADRB2 4825/4885HIF1A 3211/4885
US-11312704-B2 Inhibitors of cysteine proteases and methods of use thereof CTSV, CTRL, CTSL ADRB1 4867/4885ADRB2 4846/4885HIF1A 3242/4885
US-20220324875-A1 CHEMICAL COMPOUNDS PIK3CA, PIK3CD, PIK3CB ADRB1 2903/4885ADRB2 3588/4885HIF1A 3161/4885
US-20250084077-A1 ETHER LINKED TRIAZOLES AS NRF2 ACTIVATORS NFE2L2, KEAP1, NQO1 ADRB1 871/4885ADRB2 965/4885HIF1A 439/4885
US-20220204526-A1 HYDROXYPYRIDOXAZEPINES AS NRF2 ACTIVATORS KEAP1, NFE2L2, NQO1 ADRB1 97/4885ADRB2 57/4885HIF1A 869/4885
US-20220162194-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTSV, CTRL, CTSL ADRB1 4867/4885ADRB2 4846/4885HIF1A 3242/4885
US-11472793-B2 Inhibitors of cysteine proteases and methods of use thereof CTSV, CTRL, CTSL ADRB1 4867/4885ADRB2 4846/4885HIF1A 3242/4885
US-20250313573-A1 HYDROXYPYRIDOXAZEPINES AS NRF2 ACTIVATORS KEAP1, NFE2L2, NQO1 ADRB1 97/4885ADRB2 57/4885HIF1A 869/4885
US-20220324844-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTSV, CTRL, CTSL ADRB1 4867/4885ADRB2 4846/4885HIF1A 3242/4885
US-11229623-B2 TRPV4 antagonists TRPV4, TRPV5, TRPV2 ADRB1 1180/4885ADRB2 1126/4885HIF1A 1995/4885
US-20250084075-A1 THERAPEUTIC COMPOUNDS NFE2L2, KEAP1, NQO1 ADRB1 708/4885ADRB2 1086/4885HIF1A 145/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.