Etoricoxib

Etoricoxib

SCHEMBL29366203

Cc1ccc(-c2ncc(Cl)cc2-c2ccc(S(C)(=O)=O)cc2)cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS2

The experimentally established mechanism targets of Etoricoxib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 20/20 1.00
PTGS1 P23219 10/20 1.00
ABCC4 O15439 1/20 1.00
ABCB11 O95342 1/20 1.00
PDE4D Q08499 1/20 1.00
MAPK14 Q16539 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etoricoxib SCHEMBL4680 1.00 PTGS2 (1.00) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL29402456 1.00 PTGS2 (1.00) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL30988052 1.00 PTGS2 (1.00) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL14163961 1.00 PTGS2 (1.00) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL183950 0.99 PTGS2 (0.97) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL321747 0.99 PTGS2 (0.97) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL28893910 0.99 PTGS2 (0.97) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL14126237 0.99 PTGS2 (0.97) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL322344 0.99 PTGS2 (0.97) PTGS2PTGS1ABCC4ABCB11PDE4D
Etoricoxib SCHEMBL28319282 0.97 PTGS2 (0.95) PTGS2PTGS1ABCC4ABCB11PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 201 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118647367-A Novel injectable combination formulations 南爱克萨股份公司 2024-09-13 CN claimed
CN-115806521-A Monofluoromethyl etoricoxib and preparation method thereof 华东理工大学 2023-03-17 CN claimed
CN-115209880-A Nanoparticles for treating eye diseases 雷根斯堡大学 2022-10-18 CN claimed
US-20260144674-A1 Apparatus and Methods for Drug Delivery Using Microneedles CLEARSIDE BIOMEDICAL, INC. (US) 2026-05-28 US disclosed
CN-116209679-B Antibody-drug conjugates containing anti-mesothelin antibodies and uses thereof BIOTECHNOLOGY DEVELOPMENT CENTER (CN) 2026-05-26 CN disclosed
EP-3509604-B1 COMBINATION THERAPIES USING IMMUNO-DASH INHIBITORS AND PGE2 ANTAGONISTS TUFTS COLLEGE (US) 2026-02-18 EP disclosed
US-12545750-B2 Method for the diimide hydrogenation of emulsified unsaturated polymers PARKER DANE K (US) 2026-02-10 US disclosed
EP-4682148-A2 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES AbbVie Ireland Unlimited Company (IE) 2026-01-21 EP disclosed
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors CARDURION PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
US-12508227-B2 Dry powder compositions with magnesium stearate Aspeya US Inc. (US) 2025-12-30 US disclosed
US-20250368786-A1 NOVEL SARGASSUM-BASED POLYMER COMPOSITE FILAMENTS FOR 3D PRINTING AND METHOD OF MAKING THE SAME POLYTECHNIC UNIVERSITY OF PUERTO RICO 2025-12-04 US disclosed
US-20220098207-A1 FUSED HETEROARYL COMPOUNDS AND THEIR USE AS CAMKII INHIBITORS CARDURION PHARMACEUTICALS, INC. 2022-03-31 US disclosed
CN-114246953-A anti-cMet antibody drug conjugates and methods of use thereof 艾伯维生物制药股份有限公司 2022-03-29 CN disclosed
CN-114245807-A FLT3L-FC fusion proteins and methods of use 吉利德科学公司 2022-03-25 CN disclosed
CN-114222582-A Peptides and uses thereof 横向知识产权私人有限公司 2022-03-22 CN disclosed
US-20220081445-A1 CYCLIC MOLECULES AS BRUTON'S TYROSINE KINASE INHIBITOR MINGHUI PHARMACEUTICAL SHANGHAI LTD (CN) 2022-03-17 US disclosed
CN-114177308-A anti-cMet antibody drug conjugates and methods of use thereof 艾伯维生物制药股份有限公司 2022-03-15 CN disclosed
US-20220040149-A1 COMBINATION THERAPIES USING IMMUNO-DASH INHIBITORS AND PGE2 ANTAGONISTS TRUSTEES OF TUFTS COLLEGE 2022-02-10 US disclosed
US-20220040206-A1 DRY POWDER FORMULATIONS FOR INHALATION OTITOPIC INC (US) 2022-02-10 US disclosed
CN-110177527-B Device and method for adjusting insertion depth of needle for medicament delivery 科尼尔赛德生物医学公司 2022-02-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors RYR2, CACNA1C, CAMK4 PTGS2 1343/4885PTGS1 1270/4885ABCC4 2586/4885
US-12508227-B2 Dry powder compositions with magnesium stearate ACMSD, SARAF, TMCO1 PTGS2 26/4885PTGS1 55/4885ABCC4 1350/4885
US-20220098207-A1 FUSED HETEROARYL COMPOUNDS AND THEIR USE AS CAMKII INHIBITORS CAMK2B, CAMK2A, CAMK2G PTGS2 1154/4885PTGS1 1446/4885ABCC4 4037/4885
US-20260144674-A1 Apparatus and Methods for Drug Delivery Using Microneedles PROKR2, SLC10A2, GLP1R PTGS2 2731/4885PTGS1 3480/4885ABCC4 3092/4885
US-20220040149-A1 COMBINATION THERAPIES USING IMMUNO-DASH INHIBITORS AND PGE2 ANTAGONISTS HPGDS, PTGIS, PTGDR2 PTGS2 19/4885PTGS1 16/4885ABCC4 3747/4885
US-12545750-B2 Method for the diimide hydrogenation of emulsified unsaturated polymers ALOX15, SOD1, ALOX12 PTGS2 188/4885PTGS1 459/4885ABCC4 578/4885
US-20220081445-A1 CYCLIC MOLECULES AS BRUTON'S TYROSINE KINASE INHIBITOR ABL1, BTK, LYN PTGS2 3974/4885PTGS1 3564/4885ABCC4 3642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.