Sulisobenzone

Sulisobenzone

SCHEMBL29378407

COc1cc(O)c(C(=O)c2ccccc2)cc1S(=O)(=O)[O-].[Na+]

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Sulisobenzone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A known ✓ P27815 1/20 0.51
PDE4D known ✓ Q08499 1/20 0.51
PTGS1 known ✓ P23219 1/20 0.41
PTGS2 known ✓ P35354 1/20 0.41
NOD2 known ✓ Q9HC29 1/20 0.40
LMNA P02545 5/20 0.76
MAPT P10636 5/20 0.76
KMT2A Q03164 4/20 0.76
ALDH1A1 P00352 3/20 0.76
HPGD P15428 3/20 0.66
KDM4E B2RXH2 2/20 0.66
HSD17B10 Q99714 2/20 0.66
CYP3A4 P08684 1/20 0.66
RECQL P46063 1/20 0.66
HTT P42858 3/20 0.51
MAPK1 P28482 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C19 P33261 2/20 0.51
PGR P06401 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulisobenzone SCHEMBL338882 1.00 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL28588923 0.99 LMNA (0.74) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL11277588 0.97 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL6295947 0.97 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL10621756 0.97 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL10491696 0.97 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL10723288 0.97 LMNA (0.76) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL2209368 0.94 LMNA (0.71) LMNAMAPTKMT2AALDH1A1HPGD
Sulisobenzone SCHEMBL5147287 0.90 LMNA (0.65) LMNAMAPTKMT2AALDH1A1HPGD
SCHEMBL240880 0.87 LMNA (0.56) LMNAMAPTKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 122 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3600224-B1 SKIN CARE COMPOSITIONS COMPRISING A TERPOLYMER, PROCESS FOR PREPARING THE SAME AND METHOD OF USE THEREOF ISP INVESTMENTS LLC (US) 2026-05-06 EP claimed
EP-4518849-B1 COMPOSITION FOR TOPICAL APPLICATION FOR THE PHOTOTHERAPEUTIC TREATMENT OF INFLAMMATORY-BASED SKIN DISEASES GIULIANI SPA (IT) 2026-04-08 EP claimed
EP-3709966-B1 COMPOSITIONS COMPRISING AT LEAST ONE ACRYLIC POLYMER AND AT LEAST ONE INSOLUBLE ORGANIC SCREENING AGENT OREAL (FR) 2024-12-11 EP claimed
WO-2024027193-A1 SKIN-CARE PRODUCT COMPOSITION AND PHARMACEUTICAL COMPOSITION COMPRISING SULFONATED CALIXARENE, AND USE OF SULFONATED CALIXARENE 苏州隽德生物科技有限公司 2024-02-08 WO claimed
CN-113754932-B Photo-aging-resistant latex product and manufacturing method thereof 温州卡美琳乳胶制品有限公司 2023-03-03 CN claimed
CN-115003388-A Aqueous sunscreen formulations based on sulfated crystalline cellulose SPF boosters 陶氏环球技术有限责任公司 2022-09-02 CN claimed
EP-3773444-B1 COSMETIC COMPOSITION FOR A FAST SWEAT EVAPORATION BEIERSDORF AG (DE) 2022-03-02 EP claimed
CN-108671267-B Absorbent and reflective biocompatible dyes for high precision medical implants H·戴维·迪恩 2022-02-18 CN claimed
EP-3946642-A1 SUNSCREEN COMPOSITIONS AND METHOD OF USE THEREOF ISP Investments LLC (US) 2022-02-09 EP claimed
EP-3600224-B1 SKIN CARE COMPOSITIONS COMPRISING A TERPOLYMER, PROCESS FOR PREPARING THE SAME AND METHOD OF USE THEREOF ISP INVESTMENTS LLC (US) 2026-05-06 EP disclosed
EP-4104010-B1 A FUNCTIONAL AND TRANSPARENT GEL ELECTROLYTE SYSTEM AND FAST SWITCHING ELECTROCHROMIC/ELECTROCHEMICAL DEVICES THEREOF COUNCIL OF SCIENT AND INDUSTRIAL RESEARCH AN INDIAN REGISTERED BODY INCORPORATED UNDER REGN OF SOC A (IN) 2026-05-06 EP disclosed
EP-3389618-B2 PROCESS FOR TREATING KERATIN FIBRES USING AN AQUEOUS COMPOSITION COMPRISING A COMBINATION OF PARTICULAR ALKOXYSILANES OREAL (FR) 2026-04-22 EP disclosed
WO-2026044006-A1 MODIFIED STARCH COMPOUNDS AND USES THEREOF ISP INVESTMENTS LLC (US) 2026-02-26 WO disclosed
EP-4698227-A1 SUPRAMOLECULAR ASSEMBLIES, COMPOSITIONS COMPRISING THE SAME AND METHODS FOR PRODUCING THE SAME ELC Management LLC (US) 2026-02-25 EP disclosed
CN-110785452-B Process for preparing organopolysiloxane gels 瓦克化学股份公司 2022-05-13 CN disclosed
US-20220144785-A1 COMPOUNDS HAVING EXCITED STATE INTRAMOLECULAR PROTON TRANSFER (ESIPT) CHARACTER FOR USE IN TREATING AND/OR PREVENTING SUNBURN AND/OR PREVENTING U.V. DAMAGE UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2022-05-12 US disclosed
WO-2022063405-A1 METHOD FOR PRODUCING HYDROPHILIC ORGANOPOLYSILOXANE GELS WACKER CHEMIE AG (DE) 2022-03-31 WO disclosed
CN-109475482-B Medicine 西姆莱斯股份公司 2022-03-29 CN disclosed
CN-114206426-A Device and method for applying a cosmetic composition by means of a grated end-effector 强生消费者公司 2022-03-18 CN disclosed
CN-108671267-B Absorbent and reflective biocompatible dyes for high precision medical implants H·戴维·迪恩 2022-02-18 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220144785-A1 COMPOUNDS HAVING EXCITED STATE INTRAMOLECULAR PROTON TRANSFER (ESIPT) CHARACTER FOR USE IN TREATING AND/OR PREVENTING SUNBURN AND/OR PREVENTING U.V. DAMAGE NNT, NQO1, SUN2 PDE4A 4862/4885PDE4D 4815/4885PTGS1 1801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.