Primaperone

Primaperone

SCHEMBL310299

O=C(CCCN1CCCCC1)c1ccc(F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.74
HTR1A P08908 5/20 0.70
DRD3 P35462 5/20 0.70
DRD1 P21728 3/20 0.70
ADRA2A P08913 2/20 0.70
ADRA1A P35348 2/20 0.70
OPRM1 P35372 2/20 0.70
KCNH2 Q12809 2/20 0.70
HRH3 Q9Y5N1 2/20 0.70
MEN1 O00255 1/20 0.70
CHRM2 P08172 1/20 0.70
KMT2A Q03164 1/20 0.70
SLC6A4 P31645 2/20 0.69
SLC6A3 Q01959 2/20 0.69
DRD2 P14416 6/20 0.67
DRD4 P21917 3/20 0.65
HTR2A P28223 3/20 0.65
HTR2C P28335 3/20 0.65
HRH1 P35367 3/20 0.65
TMEM97 Q5BJF2 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Primaperone SCHEMBL364809 0.98 TSHR (0.76) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL4496558 0.98 TSHR (0.76) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL11755100 0.90 ALDH1A1 (0.71) TSHRHTR1AADRA1AKCNH2HRH3
Primaperone SCHEMBL30110541 0.90 TSHR (0.68) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL7350313 0.89 ALDH1A1 (0.68) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL11790502 0.87 HTR1A (0.69) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL7375822 0.87 HRH3 (0.58) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL7378554 0.87 HRH3 (0.58) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL28432024 0.86 TSHR (0.72) TSHRHTR1ADRD3DRD1ADRA2A
SCHEMBL16986166 0.86 TSHR (0.97) TSHRHTR1ADRD3DRD1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 420 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20020115655-A1 Such as S-(4-methoxybenzyl)-N-(2-(N',N'-dimethylamino)ethyl) thiosalicylamide; for treatment of cardiovascular disorders MASSACHUSETTS COLLEGE OF PHARMACY 2002-08-22 US claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-12605384-B2 Uses INTRA-CELLULAR THERAPIES, INC. (US) 2026-04-21 US disclosed
EP-3746081-B1 PDE1 INHIBITORS FOR USE TO TREAT CARDIAC FAILURE AND CARDIOTOXICITY INTRA CELLULAR THERAPIES INC (US) 2026-04-01 EP disclosed
US-20260049314-A1 ANTISENSE OLIGONUCLEOTIDE-BASED ANTI-FIBROTIC THERAPEUTICS UNIVERSITY OF ROCHESTER (US) 2026-02-19 US disclosed
EP-4581143-A1 ANTISENSE OLIGONUCLEOTIDE-BASED ANTI-FIBROTIC THERAPEUTICS University of Rochester (US) 2025-07-09 EP disclosed
US-20250066790-A1 ANTISENSE OLIGONUCLEOTIDES FOR MODIFYING PROTEIN EXPRESSION UNIVERSITY OF ROCHESTER 2025-02-27 US disclosed
US-20250018009-A1 SERUM RESPONSE FACTOR REGENERATES SENESCENT CELLS UNIVERSITY OF HOUSTON SYSTEM (US) 2025-01-16 US disclosed
EP-0737066-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1996-10-16 EP disclosed
US-5446070-A Flexible, finite, bioadhesive, therapeutical agent in solid form NOVER PHARMACEUTICALS, INC. (US) 1995-08-29 US disclosed
WO-1995018603-A1 TRANSDERMAL DEVICE CONTAINING POLYVINYLPYRROLIDONE AS SOLUBILITY ENHANCER NOVEN PHARMACEUTICALS, INC. (US) 1995-07-13 WO disclosed
US-4772616-A DOMPERIDONE THE TEXAS A & M UNIVERSITY SYSTEM (US) 1988-09-20 US disclosed
US-4284638-A Pharmaceutical compositions with central depressant and antipsychotic activity having a butyrophenone derivative which is substituted in the 4-position and a C-(2-benzofuranyl)-piperidine or C-(2-benzofuranyl)-tetrahydro-pyridine CIBA-GEIGY CORPORATION (US) 1981-08-18 US disclosed
US-3936468-A PSYCHOTROPIC SUMITOMO CHEMICAL COMPANY, LTD. (JA) 1976-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260049314-A1 ANTISENSE OLIGONUCLEOTIDE-BASED ANTI-FIBROTIC THERAPEUTICS UPF1, HNRNPF, RNMT TSHR 2997/4885HTR1A 3926/4885DRD3 4661/4885
US-20020115655-A1 Such as S-(4-methoxybenzyl)-N-(2-(N',N'-dimethylamino)ethyl) thiosalicylamide; for treatment of cardiovascular disorders CACNA1G, CACNA1F, CACNA1H TSHR 4456/4885HTR1A 660/4885DRD3 3204/4885
US-12605384-B2 Uses PDE2A, NPR1, PDE7A TSHR 105/4885HTR1A 228/4885DRD3 1392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.