SCHEMBL366741

SCHEMBL366741

NC(=O)c1c2ccccc2n2cc(S(=O)(=O)C3CC3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.38
SRC P12931 1/20 0.38
HTR2A P28223 5/20 0.36
HTR2C P28335 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CCR6 P51684 3/20 0.34
HTR3A P46098 1/20 0.34
KCNH2 Q12809 3/20 0.32
DRD2 P14416 2/20 0.32
CCR7 P32248 1/20 0.32
SPR P35270 1/20 0.32
NPC1 O15118 1/20 0.32
AGTR1 P30556 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C1 Q04828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365147 0.90 AGTR1 (0.39) EGFRHTR2AHTR2CMEN1KMT2A
SCHEMBL364653 0.82 CA2 (0.43) EGFRSRCHTR2AHTR2CAGTR1
SCHEMBL367707 0.81 EGFR (0.44) EGFRSRCHTR2AHTR2CMEN1
SCHEMBL366740 0.80 KDM4E (0.36) EGFRSRCHTR2AHTR2CMEN1
SCHEMBL366999 0.78 EGFR (0.42) EGFRSRCMEN1KMT2A
SCHEMBL366926 0.77 ALDH1A1 (0.36) EGFRSRCHTR2AHTR2CMEN1
SCHEMBL367201 0.75 EGFR (0.45) EGFRSRCHTR2AHTR2CAGTR1
SCHEMBL367764 0.75 EGFR (0.45) EGFRSRCHTR2AHTR2CMEN1
SCHEMBL365648 0.73 CA9 (0.45) EGFRAGTR1CA12CA1CA2
SCHEMBL365259 0.72 KDM4E (0.44) EGFRSRCHTR2AHTR2CAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed