SCHEMBL367616

SCHEMBL367616

COC(=O)c1c2ccccc2n2cc(OC(=O)N(C)C)cc(O)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 5/20 0.46
NR4A2 P43354 3/20 0.40
KMT2A Q03164 4/20 0.38
MEN1 O00255 1/20 0.38
PKM P14618 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.37
SRC P12931 2/20 0.37
EGFR P00533 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365213 0.89 PKM (0.39) NCEH1KMT2AMEN1PKMALDH1A1
SCHEMBL365256 0.88 EGFR (0.40) NCEH1KMT2AMEN1PKMALDH1A1
SCHEMBL367734 0.78 ATM (0.40) NCEH1KMT2AMEN1PKMALDH1A1
SCHEMBL365490 0.77 NCEH1 (0.39) NCEH1KMT2AMEN1PKMSRC
SCHEMBL367615 0.73 IDO1 (0.42) NCEH1KMT2AMEN1PKMALDH1A1
SCHEMBL366828 0.72 PKM (0.46) NCEH1KMT2APKMALDH1A1SRC
SCHEMBL367283 0.71 RAB9A (0.44) NCEH1KMT2APKMALDH1A1SRC
SCHEMBL365189 0.70 ACHE (0.37) NCEH1ALDH1A1
SCHEMBL365769 0.70 LTB4R (0.39) KMT2AMEN1PKMALDH1A1KDM4E
SCHEMBL364802 0.70 KDM4E (0.49) KMT2AMEN1PKMALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed