SCHEMBL367175

SCHEMBL367175

CN(C)CCc1cc2c(C(=O)O)c3ccccn3c2cc1C(=O)N(C)C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 8/20 0.39
HTR6 P50406 12/20 0.38
PTGS2 P35354 1/20 0.38
HTR1A P08908 4/20 0.38
HTR1D P28221 4/20 0.38
HTR1B P28222 4/20 0.38
HTR1F P30939 4/20 0.38
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
TACR1 P25103 1/20 0.37
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367176 0.78 HTR6 (0.38) HTR7HTR6PTGS2HTR1AHTR1D
SCHEMBL367174 0.77 IDO1 (0.37) PTGS2TACR1ALDH1A1IDO1
SCHEMBL367204 0.74 RORC (0.43) PTGS2TACR1ALDH1A1IDO1
SCHEMBL366132 0.70 ALDH1A1 (0.38) HTR7HTR6PTGS2HTR1AHTR1D
SCHEMBL366535 0.70 EGFR (0.48) ALDH1A1IDO1
SCHEMBL366827 0.67 KMT2A (0.45) ALDH1A1CYP1A2POLB
SCHEMBL365387 0.67 ALDH1A1 (0.46) ALDH1A1CYP1A2POLB
SCHEMBL371112 0.67 IDO1 (0.51) PTGS2TACR1ALDH1A1CYP1A2POLB
SCHEMBL366461 0.66 HTT (0.46) PTGS2ALDH1A1IDO1
SCHEMBL366789 0.65 IDO1 (0.38) PTGS2TACR1ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed