SCHEMBL3974894

SCHEMBL3974894

COc1cc2c(c(Br)c1OC)CN(CCN1CCCCC1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.44
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
HTR4 Q13639 1/20 0.39
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
HTR2C P28335 2/20 0.38
ATM Q13315 1/20 0.38
MEN1 O00255 1/20 0.37
ABCC4 O15439 1/20 0.37
LMNA P02545 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CHRM3 P20309 1/20 0.37
MAPK1 P28482 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973213 0.99 HTR2A (0.42) HTR2APOLBSMN1; SMN2HTR4KDR
SCHEMBL4084541 0.89 SYK (0.45) SMN1; SMN2KDRLMNACYP2D6TSHR
SCHEMBL4081651 0.84 LMNA (0.46) DRD2DRD3LMNACYP2D6CYP2C9
SCHEMBL3973494 0.83 IDH1 (0.39) POLBSMN1; SMN2MEN1CYP3A4TSHR
SCHEMBL3972272 0.81 CA1 (0.38) ACHE
SCHEMBL3973824 0.81 HTR2A (0.36) HTR2ASMN1; SMN2KDRDRD2
SCHEMBL3979633 0.81 POLB (0.43) POLBSMN1; SMN2DRD2DRD3MEN1
SCHEMBL3971360 0.79 ALDH1A1 (0.43) KDRMEN1CYP3A4CYP2D6THPO
SCHEMBL3973796 0.79 HSD17B10 (0.46) SMN1; SMN2HTR2CCYP2D6CYP2C9TSHR
SCHEMBL3973411 0.78 CNR2 (0.45) KCNH2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009051417-A2 PHENANTHRENE LACTAM DERIVATIVES HAVING ANTICANCER ACTIVITY AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-04-23 WO disclosed