SCHEMBL4041149

SCHEMBL4041149

COc1ccc(CC(NC(=O)Oc2ccc(-c3ccccc3)cc2)C(=O)N2CCC3C2C(=O)CN3C(=O)Cc2cccnc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 7/20 0.39
ITGB7 P26010 7/20 0.39
CTSK P43235 2/20 0.39
KLKB1 P03952 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
F2 P00734 2/20 0.38
MAPT P10636 1/20 0.37
ECE1 P42892 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CHRNA7 P36544 1/20 0.36
MMP12 P39900 1/20 0.36
ACE P12821 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049549 0.94 GPR132 (0.38) ITGA4ITGB7CTSKECE1CHRNA7
SCHEMBL4040214 0.93 GPR132 (0.39) ITGA4ITGB7CTSKKLKB1ECE1
SCHEMBL4045083 0.90 CTSK (0.47) CTSKCHRNA7
SCHEMBL4042165 0.90 EPHX1 (0.37) CTSKECE1CHRNA7ACE
SCHEMBL4047771 0.89 CTSK (0.39) CTSKECE1CHRNA7
SCHEMBL4045511 0.87 F2 (0.38) ITGA4ITGB7CTSKITGB3ITGAV
SCHEMBL4044931 0.85 CTSK (0.54) CTSKF2MAPTALDH1A1GAA
SCHEMBL4042585 0.84 USP30 (0.39) ITGA4ITGB7CTSKITGB3ITGAV
SCHEMBL4041556 0.84 CTSK (0.43) ITGA4ITGB7CTSKITGB3ITGAV
SCHEMBL4043904 0.84 DPP4 (0.44) F2MAPTALDH1A1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed