SCHEMBL4040214

SCHEMBL4040214

O=C(NC(Cc1ccc(F)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 2/20 0.39
SCN9A Q15858 1/20 0.38
CTSK P43235 2/20 0.37
MC4R P32245 1/20 0.37
MC3R P41968 1/20 0.37
MC1R Q01726 1/20 0.37
ECE1 P42892 1/20 0.37
CHRNA7 P36544 1/20 0.36
ACE P12821 2/20 0.36
ITGA4 P13612 2/20 0.36
ITGB7 P26010 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
GPR34 Q9UPC5 1/20 0.36
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PRCP P42785 1/20 0.35
PSMB5 P28074 1/20 0.35
KLKB1 P03952 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049549 0.94 GPR132 (0.38) GPR132CTSKECE1CHRNA7ACE
SCHEMBL4041149 0.93 ITGA4 (0.39) CTSKECE1CHRNA7ACEITGA4
SCHEMBL4042165 0.90 EPHX1 (0.37) GPR132CTSKECE1CHRNA7ACE
SCHEMBL4045083 0.89 CTSK (0.47) CTSKCHRNA7
SCHEMBL4047771 0.88 CTSK (0.39) GPR132CTSKECE1CHRNA7
SCHEMBL4050328 0.87 SCN9A (0.39) GPR132SCN9ACTSKMC4RMC3R
SCHEMBL4041436 0.85 ALDH1A1 (0.39) GPR132SCN9AMC4RMC3RMC1R
SCHEMBL4043465 0.84 MC4R (0.41) GPR132SCN9ACTSKMC4RMC3R
SCHEMBL4052754 0.84 CTSK (0.42) SCN9ACTSKMC4RMC3RMC1R
SCHEMBL4046533 0.83 MAPK1 (0.36) GPR132CTSKMC4RMC3RMC1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed