SCHEMBL4044339

SCHEMBL4044339

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
CTSK P43235 3/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
MC4R P32245 1/20 0.33
MC3R P41968 1/20 0.33
MC1R Q01726 1/20 0.33
ALOX5 P09917 1/20 0.33
GPR132 Q9UNW8 3/20 0.32
NR2F2 P24468 2/20 0.32
RAB9A P51151 2/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
ELANE P08246 1/20 0.32
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051965 0.94 MC4R (0.38) ALDH1A1CTSKMC4RMC3RMC1R
SCHEMBL4039893 0.93 CTSK (0.41) ALDH1A1CTSKPREPFAPRAB9A
SCHEMBL4046989 0.90 ALDH1A1 (0.38) ALDH1A1PPARGPPARAPREPFAP
SCHEMBL4043678 0.90 ALDH1A1 (0.38) ALDH1A1CTSKPPARGPPARAPREP
SCHEMBL4047431 0.89 ALDH1A1 (0.37) ALDH1A1PPARGPPARAPREPFAP
SCHEMBL4043596 0.88 ELANE (0.38) ALDH1A1CTSKPREPFAPMC4R
SCHEMBL4043124 0.87 POLB (0.34) ALDH1A1CTSKRAB9AELANELMNA
SCHEMBL4043183 0.86 CTSK (0.43) ALDH1A1CTSKPREPFAPMC4R
SCHEMBL4046799 0.86 ALDH1A1 (0.39) ALDH1A1CTSKPREPFAP
SCHEMBL4045687 0.86 MC4R (0.34) ALDH1A1CTSKPREPFAPMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed