SCHEMBL4050328

SCHEMBL4050328

O=C(NC(Cc1ccc(F)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.39
GPR132 Q9UNW8 2/20 0.38
MC4R P32245 1/20 0.37
MC3R P41968 1/20 0.37
MC1R Q01726 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
P2RX7 Q99572 2/20 0.36
PSMB5 P28074 1/20 0.35
FKBP1A P62942 1/20 0.35
F2 P00734 1/20 0.35
CHRNA7 P36544 1/20 0.35
ACE P12821 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047615 0.94 CTSB (0.38) GPR132TAAR1CTSBCTSSCTSK
SCHEMBL4045511 0.93 F2 (0.38) CTSBCTSSCTSKF2ITGA4
SCHEMBL4041436 0.91 ALDH1A1 (0.39) SCN9AGPR132MC4RMC3RMC1R
SCHEMBL4044160 0.90 CTSB (0.37) SCN9AGPR132TAAR1CTSBCTSS
SCHEMBL4043952 0.89 CTSK (0.42) CTSBCTSSCTSKFKBP1ACHRNA7
SCHEMBL4043465 0.89 MC4R (0.41) SCN9AGPR132MC4RMC3RMC1R
SCHEMBL4049324 0.89 MC4R (0.37) SCN9AMC4RMC3RMC1RCTSK
SCHEMBL4043998 0.89 FKBP1A (0.37) CTSBCTSSCTSKFKBP1ACHRNA7
SCHEMBL4040214 0.87 GPR132 (0.39) SCN9AGPR132MC4RMC3RMC1R
SCHEMBL4046868 0.84 ITGB1 (0.37) GPR132CTSBCTSSCTSKP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed