SCHEMBL4051785

SCHEMBL4051785

COc1ccc(CC(NC(=O)Oc2ccc(-c3ccccc3)cc2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)Cc2ccccn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 3/20 0.39
ITGB7 P26010 3/20 0.39
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
HDAC8 Q9BY41 1/20 0.36
USP30 Q70CQ3 1/20 0.36
HTRA1 Q92743 4/20 0.35
ELANE P08246 1/20 0.35
CTSK P43235 2/20 0.35
CAPN1 P07384 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.34
STS P08842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044539 0.94 ITGA4 (0.36) ITGA4ITGB7HDAC8ELANECTSK
SCHEMBL4049324 0.93 MC4R (0.37) ITGA4ITGB7ITGB3ITGAVELANE
SCHEMBL4045311 0.90 CTSK (0.43) MMP1MMP2MMP3MMP7MMP9
SCHEMBL4046932 0.89 GPR132 (0.35) ITGA4ITGB7ITGB3ITGAVHDAC8
SCHEMBL4043139 0.89 ELANE (0.37) ITGA4ITGB7MMP1MMP2MMP3
SCHEMBL4045511 0.89 F2 (0.38) ITGA4ITGB7MMP8MMP13ITGB3
SCHEMBL4045924 0.88 USP30 (0.40) ITGA4ITGB7ITGB3ITGAVHDAC8
SCHEMBL4039691 0.86 CTSK (0.50) USP30HTRA1CTSKALDH1A1STS
SCHEMBL4038911 0.85 DPP4 (0.43) HDAC8ALDH1A1GAASTS
SCHEMBL4041003 0.85 CTSL (0.39) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed