SCHEMBL434790

SCHEMBL434790

CS(=O)(=O)NCc1ccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.47
OPRD1 P41143 3/20 0.47
OPRK1 P41145 3/20 0.47
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
CCR3 P51677 1/20 0.41
CYP2D6 P10635 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
OPRL1 P41146 1/20 0.41
P2RX7 Q99572 1/20 0.41
TRPA1 O75762 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433833 0.91 OPRM1 (0.47) OPRM1OPRD1OPRK1ALDH1A1MEN1
SCHEMBL435467 0.87 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AKDM4EPOLB
Hydrochloric Acid SCHEMBL433923 0.84 HSD11B1 (0.49) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL433860 0.82 P2RX7 (0.55) CYP2D6P2RX7TRPA1
SCHEMBL435241 0.82 P2RX7 (0.42) ALDH1A1KDM4EPOLBRAB9AP2RX7
SCHEMBL435915 0.82 P2RX7 (0.60) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL433922 0.81 SMN1; SMN2 (0.53) ALDH1A1MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL433030 0.81 SLC6A3 (0.45) OPRM1OPRK1ALDH1A1MEN1KMT2A
SCHEMBL432970 0.81 CYP1A2 (0.44) ALDH1A1MEN1KMT2ASMN1; SMN2GLA
SCHEMBL435352 0.81 P2RX7 (0.43) ALDH1A1MEN1KMT2AKDM4ECCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed