SCHEMBL4405673

SCHEMBL4405673

O=C(NC1CCN(CCN2CCCCCC2)CC1)Oc1cc2c(-c3ccc(OC(F)(F)F)cc3)cccc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.42
CHRM4 P08173 2/20 0.41
MCHR1 Q99705 2/20 0.39
HRH3 Q9Y5N1 2/20 0.39
DRD4 P21917 2/20 0.38
HTR2A P28223 2/20 0.38
CXCR3 P49682 1/20 0.38
DRD2 P14416 1/20 0.38
WNT1 P04628 1/20 0.37
DYRK1A Q13627 1/20 0.37
ACP1 P24666 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
SSTR5 P35346 1/20 0.37
KCNH2 Q12809 1/20 0.36
DRD3 P35462 1/20 0.36
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406835 0.90 CHRM3 (0.40) CHRM3MCHR1DRD4DRD2WNT1
SCHEMBL4396992 0.89 KMT2A (0.41) CHRM3MCHR1DRD4DYRK1AKCNH2
SCHEMBL4396337 0.88 HTR7 (0.43)
SCHEMBL4396457 0.88 HRH3 (0.42) HRH3DRD2KCNH2
SCHEMBL4410349 0.88 HRH3 (0.42) HRH3DRD2KCNH2
SCHEMBL4396410 0.88 L3MBTL1 (0.40) MCHR1HRH3WNT1DYRK1A
SCHEMBL913892 0.87 DRD4 (0.43) CHRM3MCHR1HRH3DRD4HTR2A
SCHEMBL4401571 0.86 HPGDS (0.39) WNT1DYRK1A
SCHEMBL4394199 0.85 CHRM3 (0.41) CHRM3WNT1DYRK1A
SCHEMBL4405570 0.83 TLR7 (0.43) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed