SCHEMBL4484664

SCHEMBL4484664

CCc1c(C(=O)O)c(C=O)n(Cc2ccccc2)c1-c1cccc(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.45
CCR2 P41597 1/20 0.41
FEN1 P39748 1/20 0.41
GRIA2 P42262 1/20 0.40
GRIA4 P48058 1/20 0.40
AR P10275 1/20 0.39
SLC16A3 O15427 1/20 0.39
SLC16A1 P53985 1/20 0.39
MCTS1 Q9ULC4 1/20 0.39
F11 P03951 1/20 0.38
PIN1 Q13526 1/20 0.38
NTRK1 P04629 1/20 0.38
NTRK3 Q16288 1/20 0.38
NTRK2 Q16620 1/20 0.38
SCD O00767 1/20 0.37
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
ADORA2A P29274 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492336 0.89 AR (0.47) FEN1GRIA2GRIA4ARALDH1A1
SCHEMBL4494579 0.86 ALDH1A1 (0.43) ARALDH1A1LMNA
SCHEMBL4490747 0.85 PGR (0.43) CCR2SLC16A3MCTS1ALDH1A1LMNA
SCHEMBL4559832 0.85 TP53 (0.46) FEN1ALDH1A1LMNA
SCHEMBL4485732 0.82 KMT2A (0.47) CCR2FEN1SLC16A3SLC16A1MCTS1
SCHEMBL4477472 0.81 PGR (0.48) CFTRCCR2FEN1ARALDH1A1
SCHEMBL4493743 0.80 GRIA2 (0.39) GRIA2GRIA4ALDH1A1LMNA
SCHEMBL4485664 0.78 KDM4E (0.40) ALDH1A1LMNA
SCHEMBL4490040 0.77 GFER (0.47) FEN1ALDH1A1
SCHEMBL4504902 0.75 AR (0.57) CFTRARALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed