SCHEMBL4566581

SCHEMBL4566581

CN(C(=O)OCc1cn(S(=O)(=O)c2cccc(C#N)c2)c(-c2cccnc2C#N)c1F)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPME1 Q9Y570 3/20 0.36
RORC P51449 6/20 0.33
AOC3 Q16853 2/20 0.33
HTR6 P50406 1/20 0.33
NR3C1 P04150 1/20 0.33
NR1H3 Q13133 1/20 0.33
KAT6A Q92794 1/20 0.32
PLCG1 P19174 1/20 0.31
APLNR P35414 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2411862 0.85 RORC (0.36) PPME1RORCHTR6NR3C1NR1H3
SCHEMBL4563370 0.83 HTR6 (0.37) PPME1RORCHTR6NR3C1NR1H3
SCHEMBL2412057 0.81 PPME1 (0.34) PPME1RORCHTR6NR3C1NR1H3
SCHEMBL1580530 0.81 GLO1 (0.38) PPME1HTR6NR3C1KAT6A
Hydrochloric Acid SCHEMBL2409926 0.80 NR3C1 (0.37) PPME1HTR6NR3C1KAT6A
SCHEMBL4566599 0.80 RXFP1 (0.35) HTR6PTGDR2
SCHEMBL4566627 0.80 ABCC9 (0.33) RORCHTR6
SCHEMBL2409288 0.79 HTR6 (0.34) HTR6PLCG1PTGDR2
SCHEMBL4569945 0.79 ALDH1A1 (0.36) RORCAOC3NR1H3PTGDR2
SCHEMBL2412055 0.79 PPME1 (0.34) PPME1RORCHTR6NR3C1KAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed