SCHEMBL4703732

SCHEMBL4703732

Cc1nsc(N(CC#N)C(=O)[C@@H](N)CC(C)C)c1-c1ccc(N2CCN(CC(=O)Nc3ccccc3)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ME2 P23368 1/20 0.43
ME1 P48163 1/20 0.43
ME3 Q16798 1/20 0.43
GAA P10253 1/20 0.43
REV1 Q9UBZ9 2/20 0.43
DRD4 P21917 2/20 0.41
CETP P11597 2/20 0.41
TSHR P16473 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
HTT P42858 1/20 0.39
CA12 O43570 1/20 0.39
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
CTSL P07711 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703889 0.88 CTSS (0.37) GAAALDH1A1CTSSCTSKCTSL
SCHEMBL4702624 0.83 RORC (0.40) CTSSCTSKCTSLCTSBGFER
SCHEMBL4704763 0.83 CTSS (0.43) CTSSCTSKCTSLCTSB
SCHEMBL6235527 0.82 CTSL (0.44) CTSSCTSKCTSLCTSB
SCHEMBL4698852 0.81 CTSK (0.39) CTSSCTSKCTSLCTSB
SCHEMBL4703554 0.78 CTSS (0.51) ME2ME1ME3GAAREV1
SCHEMBL4700965 0.75 BRD4 (0.36) CTSB
SCHEMBL4699954 0.74 CTSL (0.37) ALDH1A1CA1CA2CA7CA12
SCHEMBL4701287 0.71 CTSL (0.35) CTSSCTSKCTSLCTSB
SCHEMBL4703010 0.70 CTSS (0.37) CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed