SCHEMBL4703889

SCHEMBL4703889

Cc1nsc(N(CC#N)C(=O)[C@@H](N)CC(C)C)c1-c1ccc(N2CCN(CC(N)=O)CC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.37
CTSL P07711 13/20 0.37
CTSB P07858 13/20 0.37
CTSK P43235 12/20 0.37
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
ENPP2 Q13822 1/20 0.31
SLC27A1 Q6PCB7 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702624 0.89 RORC (0.40) CTSSCTSLCTSBCTSK
SCHEMBL4703732 0.88 ME2 (0.43) CTSSCTSLCTSBCTSKGAA
SCHEMBL4704763 0.88 CTSS (0.43) CTSSCTSLCTSBCTSK
SCHEMBL6235527 0.88 CTSL (0.44) CTSSCTSLCTSBCTSK
SCHEMBL4698852 0.81 CTSK (0.39) CTSSCTSLCTSBCTSK
SCHEMBL4700965 0.80 BRD4 (0.36) CTSB
SCHEMBL4699954 0.79 CTSL (0.37) CTSSCTSLCTSBCTSKALDH1A1
SCHEMBL4701237 0.76 CTSS (0.36) CTSSCTSLCTSBCTSK
SCHEMBL4703010 0.76 CTSS (0.37) CTSSCTSLCTSBCTSK
SCHEMBL4699979 0.76 CTSS (0.44) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed