SCHEMBL4699954

SCHEMBL4699954

Cc1nsc(N(CC#N)C(=O)[C@@H](N)CC(C)C)c1-c1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.37
CTSB P07858 2/20 0.37
CTSS P25774 2/20 0.37
CTSK P43235 2/20 0.37
CA2 P00918 12/20 0.36
CA1 P00915 7/20 0.36
CA7 P43166 2/20 0.36
CA4 P22748 2/20 0.36
CA9 Q16790 5/20 0.35
PPID Q08752 1/20 0.34
CA12 O43570 4/20 0.33
CA14 Q9ULX7 1/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
CHRNA7 P36544 1/20 0.32
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698852 0.87 CTSK (0.39) CTSLCTSBCTSSCTSK
SCHEMBL4700965 0.87 BRD4 (0.36) CTSB
SCHEMBL6235527 0.81 CTSL (0.44) CTSLCTSBCTSSCTSK
SCHEMBL4702624 0.80 RORC (0.40) CTSLCTSBCTSSCTSK
SCHEMBL4704763 0.79 CTSS (0.43) CTSLCTSBCTSSCTSK
SCHEMBL4703889 0.79 CTSS (0.37) CTSLCTSBCTSSCTSKALDH1A1
SCHEMBL4704247 0.78 DPP4 (0.33)
SCHEMBL4701287 0.77 CTSL (0.35) CTSLCTSBCTSSCTSK
SCHEMBL4703732 0.74 ME2 (0.43) CTSLCTSBCTSSCTSKCA2
SCHEMBL4701995 0.74 CTSK (0.37) CTSLCTSBCTSSCTSKCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed