SCHEMBL4700965

SCHEMBL4700965

CC(=O)c1ccc(-c2c(C)nsc2N(CC#N)C(=O)[C@@H](N)CC(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
CTSB P07858 2/20 0.31
AAK1 Q2M2I8 1/20 0.30
CIT O14578 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698852 0.89 CTSK (0.39) CTSB
SCHEMBL4699954 0.87 CTSL (0.37) CTSB
SCHEMBL4702624 0.83 RORC (0.40) CTSB
SCHEMBL6235527 0.82 CTSL (0.44) CTSB
SCHEMBL4704763 0.81 CTSS (0.43) CTSB
SCHEMBL4703889 0.80 CTSS (0.37) CTSB
SCHEMBL4702315 0.79 AAK1 (0.33) CTSBAAK1CIT
SCHEMBL4704247 0.79 DPP4 (0.33)
SCHEMBL4701287 0.76 CTSL (0.35) CTSB
SCHEMBL4703732 0.75 ME2 (0.43) CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed