SCHEMBL5043850

SCHEMBL5043850

CCCCNC(=O)Oc1cc(-c2csc(-c3ccccc3F)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 2/20 0.41
FAAH O00519 3/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
PLA2G4A P47712 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
GNRHR P30968 2/20 0.35
CTSK P43235 1/20 0.35
LMNA P02545 1/20 0.35
HTR1A P08908 2/20 0.34
ALOX5 P09917 1/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
SLC6A4 P31645 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5040330 0.89 NTMT1 (0.40) NCEH1FAAHCNR1CNR2PLA2G4A
SCHEMBL5044496 0.88 ATP4A (0.37) CTSKLMNAALOX5
SCHEMBL5047187 0.88 HDAC3 (0.36) CTSKALDH1A1HSD17B10
SCHEMBL5047889 0.87 MGLL (0.36) CTSKLMNAALOX5HTR2AHTR2C
SCHEMBL5044961 0.87 HTR2A (0.46) CNR1PIK3CDPIK3CAGNRHRLMNA
SCHEMBL5047174 0.87 CNR1 (0.40) CNR1CNR2HTR2AHTR2CSLC6A4
SCHEMBL5044102 0.86 MAPT (0.40) CNR1HTR2AHTR2CSLC6A4ALDH1A1
SCHEMBL5048696 0.86 CDC25A (0.43) FAAHLMNAALDH1A1
SCHEMBL5047653 0.85 ATP4A (0.38)
SCHEMBL5040295 0.84 DNM1L (0.36) FAAHCTSKALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed