SCHEMBL507649

SCHEMBL507649

CS(=O)(=O)c1ccc(OBOc2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.48
PTGS2 P35354 9/20 0.44
PTGS1 P23219 3/20 0.44
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10052767 0.83 ENPP2 (0.50) ENPP2PTGS2PTGS1PKM
SCHEMBL2349931 0.78 PSIP1 (0.50) PKM
SCHEMBL11547843 0.78 HTT (0.58) ENPP2PTGS2PTGS1
SCHEMBL1695070 0.77 ALDH1A1 (0.64) PTGS2
SCHEMBL2376239 0.77 ENPP2 (0.72) ENPP2PTGS2
SCHEMBL4050348 0.77 SMN1; SMN2 (0.68) PKM
SCHEMBL14331939 0.77 MMP13 (0.38) PKM
SCHEMBL11986371 0.76 PKM (0.70) PTGS2PTGS1PKM
SCHEMBL280156 0.76 PKM (0.70) PTGS2PTGS1PKM
SCHEMBL934211 0.75 DDB1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 317 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115835909-B Cannabinoid receptor type 2 (CB 2) modulators and uses thereof 泰昂治疗公司 2026-05-15 CN disclosed
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
CN-119013265-A GLUT9 heterocyclic inhibitors for the treatment of disease 爱尔兰好利恩治疗有限公司 2024-11-22 CN disclosed
CN-118702608-A Novel synthesis method of eremophilone 重庆圣华曦药业股份有限公司 2024-09-27 CN disclosed
CN-118324767-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-07-12 CN disclosed
CN-113999180-B Quinazoline compound, intermediate, preparation method, pharmaceutical composition and application 上海医药集团股份有限公司 2024-03-26 CN disclosed
CN-117736207-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
CN-115362003-B Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
CN-117500496-A Pyrimidine and pyridinamine compounds and their use in the treatment of diseases 艾匹根生物技术有限公司 2024-02-02 CN disclosed
CN-117396472-A SOS1 inhibitors and uses thereof 上海齐鲁锐格医药研发有限公司 2024-01-12 CN disclosed
WO-2004000811-A1 ARYLSULFONYLHYDROXAMIC ACID AND AMIDE DERIVATIVES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-12-31 WO disclosed
EP-1369421-A1 Pharmaceutical compositions comprising 2,3-Diaryl-pyrazolo[1,5-B]pyridazine derivatives GLAXO GROUP LIMITED (GB) 2003-12-10 EP disclosed
US-20030225110-A1 Tetrahydroquinoline derivatives as antithrombotic agents BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-12-04 US disclosed
EP-1032575-B1 2,3-DIARYL-PYRAZOLO(1,5-B)PYRIDAZINES DERIVATIVES, THEIR PREPARATION AND THEIR USE AS CYCLOOXYGENASE 2 (COX-2) INHIBITORS GLAXO GROUP LTD (GB) 2003-07-23 EP disclosed
US-20030040517-A1 2,3-Diaryl-pyrazolo[1,5-b]pyridazines derivatives, their preparation and their use as cyclooxygenase 2 (COX-2) inhibirors SMITHKLINE BEECHAM CORPORATION 2003-02-27 US disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed
US-20030008872-A1 2,3-Diaryl-pyrazolo[1,5-B]pyridazines derivatives, their preparation and their use as cyclooxygenase 2 (COX-2) inhibitors BESWICK PAUL JOHN (GB) 2003-01-09 US disclosed
US-6451794-B1 2,3-Diaryl-pyrazolo[1,5-b]pyridazines derivatives, their preparation and their use as cyclooxygenase 2(COX-2) inhibitors SMITHKLINE BEECHAM CORPORATION 2002-09-17 US disclosed
EP-1032575-A1 2,3-DIARYL-PYRAZOLO(1,5-B)PYRIDAZINES DERIVATIVES, THEIR PREPARATION AND THEIR USE AS CYCLOOXYGENASE 2 (COX-2) INHIBITORS GLAXO GROUP LIMITED (GB) 2000-09-06 EP disclosed
WO-1999012930-A1 2,3-DIARYL-PYRAZOLO[1,5-B]PYRIDAZINES DERIVATIVES, THEIR PREPA RATION AND THEIR USE AS CYCLOOXYGENASE 2 (COX-2) INHIBITORS GLAXO GROUP LIMITED (GB) 1999-03-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225110-A1 Tetrahydroquinoline derivatives as antithrombotic agents TFPI, TFPI2, SERPINC1 ENPP2 255/4885PTGS2 680/4885PTGS1 629/4885
US-20030008872-A1 2,3-Diaryl-pyrazolo[1,5-B]pyridazines derivatives, their preparation and their use as cyclooxygenase 2 (COX-2) inhibitors PTGS1, CBR1, PTGER1 ENPP2 2037/4885PTGS2 6/4885PTGS1 1/4885
US-20030040517-A1 2,3-Diaryl-pyrazolo[1,5-b]pyridazines derivatives, their preparation and their use as cyclooxygenase 2 (COX-2) inhibirors CBR1, CRHR1, CRHR2 ENPP2 2610/4885PTGS2 17/4885PTGS1 5/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 ENPP2 2267/4885PTGS2 1423/4885PTGS1 1019/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.