SCHEMBL5325571

SCHEMBL5325571

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(Cc3noc(C(F)(F)F)n3)c2=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RAD51 Q06609 1/20 0.35
HDAC6 Q9UBN7 14/20 0.34
HDAC1 Q13547 13/20 0.34
PTGS2 P35354 3/20 0.34
HDAC4 P56524 3/20 0.34
PTGS1 P23219 2/20 0.34
HDAC8 Q9BY41 7/20 0.34
CYP2C9 P11712 1/20 0.33
HTT P42858 1/20 0.33
HDAC5 Q9UQL6 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5334344 0.82 NR1H4 (0.32) CYP2C9HTT
SCHEMBL14622464 0.80 SMN1; SMN2 (0.43) PTGS2CYP2C9HTT
SCHEMBL5325289 0.79 HSP90AA1 (0.38) RAD51HDAC6HDAC1PTGS2HDAC4
SCHEMBL5325697 0.76 RAD51 (0.40) RAD51PTGS2PTGS1CYP2C9HTT
SCHEMBL5324677 0.76 RGS4 (0.46) PTGS2PTGS1
SCHEMBL5331474 0.75 PTGS2 (0.38) PTGS2PTGS1CYP2C9HTT
SCHEMBL5297375 0.74 MEN1 (0.42) PTGS2CYP2C9HTT
SCHEMBL5330439 0.74 LMNA (0.44) CYP2C9HTT
SCHEMBL5327085 0.73 PDE10A (0.42) CYP2C9HTT
SCHEMBL5326415 0.73 NPBWR1 (0.39) PTGS2CYP2C9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed